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CH 3502 4500
CH 3502 4500

... 16. Discuss the mechanism of cleavage of ethers by HI. 17. Explain Williamson’s synthesis of ethers. 18. Discuss Norrish type-I reaction. 19. Discuss the mechanism of Wittig reaction and its uses in organic synthesis. 20. Explain Wolf-Kishner reduction with its mechanism. 21. Give any two methods o ...
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Dess-Martin Periodinane
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New aniline photocage for carboxylic acids
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Chem 30CL - Lecture 1c - UCLA Chemistry and Biochemistry
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Discodermolide



(+)-Discodermolide is a polyketide natural product found to stabilize microtubule. (+)-discodermolide was isolated by Gunasekera and his co-workers at the Harbor Branch Oceanographic Institute from the deep-sea sponge Discodermia dissoluta in 1990. (+)-Discodermolide was found to be a potent inhibitor of tumor cell growth in several MDR cancer cell lines. (+)-discodermolide also shows some unique characters, including a linear backbone structure, immunosuppressive properties both in vitro and in vivo, potent induction of an accelerated senescence phenotype, and synergistic antiproliferative activity in combination with paclitaxel. Discodermolide was recognized as one of the most potent natural promoters of tubulin assembly. A large number of efforts toward the total synthesis of (+)-discodermolide were directed by its interesting biological activities and extreme scarcity of natural sources (0.002% w/w from frozen marine sponge). The compound supply necessary for complete clinical trials cannot be met by harvesting, isolation, and purification. As of 2005, attempts at synthesis or semi-synthesis by fermentation have proven unsuccessful. As a result, all discodermolide used in preclinical studies and clinical trials has come from large-scale total synthesis.
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