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2003-2004
Pharmacology Review
of Everything
Abacavir
Antiretroviral
Nucleoside reverse transcriptase
inhibitor (NRTI)
Abciximab
Antiplatelet
Anti-GPIIb/IIIa receptor antibody
Acarbose
Oral hypoglycemic
Alpha-glucosidase inhibitor
Inhibitor of intestinal glucose
absorption
Acebutolol
Sympatholytic
1 adrenergic antagonist
Class II antiarrhytmic
Antihypertensive
Antianginal
Bronchoconstrictor
Acetaminophen
Analgesic, Antipyretic
Acetazolamide
Diuretic
Carbonic anhydrase inhibitor
Acetylcholine
Cholinomimetic
Antigluacoma
Muscle contraction (nicotinic receptor)
Activated charcoal
Antidote
Acyclovir
Antiherpes
Purine analog
Phosphorylated to inhibitor of viral
DNA polymerase
Adenosine
Antiarrhythmic
Miscellaneous
(does not fit class I-IV organization)
Adrenocorticotropin
(ACTH)
Anterior pituitary hormone
Anticonvulsant
Stimulates synthesis
and release of cortisol
Albendazole
Antihelminthic
Treatment of intestinal roundworms
Albuterol
Sympathomimetic
2 adrenergic agonist
Short acting bronchodilator
Used in asthma
Aldosterone
Adrenocorticosteroid
Mineralocorticoid
Alemtuzumab
Antineoplastic
Anti-CD52 antibody
Alendronate
Anti-osteoporesis
Bisphosphonate
Inhibitor of osteoclast-mediated
bone resorption
Alfentanil
Opioid
General anaesthetic
Intravenous anaesthetic
Allopurinol
Antigout
Antineoplastic (supporting agent)
Folic acid analogue
Xanthine oxidase inhibitor
Alteplase
Thrombolytic
Tissue plasminogen activator (tPA)
Aluminum hydroxide
Antiulcer
Antacid
Amantadine
Antiviral
Antiparkinson
Treatment of Influenza A
Inhibits replication
at the stage of uncoating
Amikacin
Aminoglycoside antibiotic
Bactericidal protein synthesis inhibitor
30S ribosome
Freezes initiation
Amiloride
Potassium sparing diuretic
Sodium channel inhibitor
Antihypertensive
Aminocaproic acid (EACA)
Procoagulant
Inhibitor of plasminogen activation
(decreases fibrinolysis)
Aminoglutethimide
Antineoplastic
Immunosuppressive
Glucocorticoid antagonist
Aromatase inhibitor
(decreases steroid synthesis)
Aminoglycosides
Antibiotics
Bactericidal protein synthesis inhibitors
30S ribosome
Freezes initiation
Aminophylline
Bronchodilator
Methylxanthine
Phosphodiesterase inhibitor
Used in asthma
Amiodarone
Class I/III antiarrhythmic
Na+ and K+ channel blocker
(inactivated channels)
Amitriptyline
Tricyclic antidepressant (TCA)
Amlodipine
Antihypertensive
Calcium channel blocker
Amoxicillin
Penicillin antibiotic
Cell wall synthesis inhibitor
Antiulcer
Amino penicillin
Inhibits peptidoglycan cross-linking
Amphetamine
Indirect sympathomimetic
Drug of abuse
ADD treatment
Stimulant
Ampicillin
Penicillin antibiotic
Cell wall synthesis inhibitor
Antiulcer
Amino penicillin
Inhibits peptidoglycan cross-linking
Amphotericin B
Antifungal
Polyene antibiotic
Binds to ergosterol and alters permeability
Systemic
Amsacrine
Antineoplastic
Miscellaneous
Amyl nitrite
Vasodilator
Antianginal
Aerosol
Anastrozole
Antineoplastic
Antiestrogen
Aromatase inhibitor
Angiotensin II
Autacoid
Vasoconstrictor
Anistreplase
Thrombolytic
Streptokinase + plasminogen
Anti-thymocyte globulin
Immunosuppressive
Anti-T cell antibody
Aprotinin
Procoagulant
Fibrinolytic inhibitor
Serine protease inhibitor (“serpin”)
Streptokinase inhibitor
Arsenicals
Melarsoprol
Tropical antiparasitic
Treatment of African
Trypanosomiasis in CNS
L-asparaginase
Antineoplastic
Protein synthesis inhibitor
Aspirin
(Acetylsalicylic acid, ASA)
NSAID (acetylsalicylate)
Analgesic, Anti-inflammatory
Antipyretic, Antiplatelet
Irreversible cyclooxygenase inhibitor
Aspart insulin
Hormone
Insulin analogue
Ultra short acting
Atenolol
Sympatholytic
1 adrenergic antagonist
Antihypertensive
Antiarrhythmic
Antianginal
Bronchoconstrictor
Atorvastatin
Antihyperlipidemic
HMG-CoA Reductase inhibitor
Atovaquone
Antimalarial
Depolarizes parasitic mitochondria
and inhibits electron transport
Atracurium
Paralytic
Paralyzes skeletal muscles
Atropine
Anticholinergic
Antimuscarinic
Treatment for bradycardia, diarrhea,
cholinesterase poisoning
Auranofin
Disease modifying
anti-rheumatic drug (DMARD)
Gold salt
Oral
Aurothioglucose
Disease modifying
anti-rheumatic drug (DMARD)
Gold salt
Parenteral
Azathioprine
Immunosuppressive
Antineoplastic
Antimetabolite
(“pseudofeedback inhibition” of
HGPRT and PRP)
Azithromycin
Macrolide antibiotic
Bacteriostatic protein synthesis inhibitor
Antiulcer
50S ribosome
Inhibits translocation
Aztreonam
New  lactam antibiotic
Monobactam
Bacitracin
Antibiotic
Cell wall synthesis inhibitor
Topical, not a  lactam,
Inhibits dephosphorylation of
bactoprenol
Baclofen
Skeletal muscle relaxant
Anxiolytic
GABAB agonist
Balsalazide
NSAID (salicylate)
Basiliximab
Immunosuppressive
Anti-CD25 (interleukin 2 receptor)
Organ transplant (antirejection)
Beclomethasone
Adrenocorticosteroid
Glucocorticoid
Anti-inflammatory steroid
Inhaled
Benazopril
Antihypertensive
Converting enzyme inhibitor
Benzathine penicillin G
Penicillin antibiotic
Cell wall synthesis inhibitor
Inhibits peptidoglycan cross-linking
Repository preparation
Benztropine
Anticholinergic
Antiparkinson
Muscarinic receptor antagonist
Betamethasone
Adrenocorticosteroid
Glucocorticoid
Anti-inflammatory steroid
Not by inhalation
Betaxolol
Sympatholytic
1 adrenergic antagonist
Antihypertensive
Glaucoma medication
Bronchoconstrictor
Bethanecol
Cholinomimetic
Muscarinic agonist
Induces defecation and urination
Bronchoconstrictor
Bicalutamide
Antiandrogen
Androgen receptor antagonist
Biltolterol
Sympathomimetic
2 adrenergic agonist
Bronchodilator
Bisacodyl
Contact cathartic
Bismuth subsalicylate
Antiulcer
Antidiarrheal
Bispropolol
Sympatholytic
 adrenergic antagonist
Antihypertensive
Bronchoconstrictor
Bivalirudin
Anticoagulant
Thrombin inhibitor
Black cohosh
Dietary supplement
Relief of “hot flashes” and other
menopausal symptoms
Bleomycin
Antineoplastic
Natural product
Antibiotic
Botulinum toxin
(Botox)
Paralytic
Paralyzes skeletal muscles
Bradykinin
Inflammatory mediator
Plasma, hypotension, pain
Bretylium
Sympatholytic
Class III antiarrhythmic
K+ channel blocker
Bromocriptine
Antiparkinson
Dopamine (D2) agonist
Inhibits prolactin release
Brupropion
Second generation antidepressant
Bumetanide
Loop diuretic
Na+-K+-2Cl- transporter inhibitor
Buprenorphine
Opioid
Partial agonist
Buspirone
Sedative/hypnotic
Anxiolytic
Busulfan
Antineoplastic
Alkylating Agent
Budenoside
Adrenocorticosteroid
Glucocorticoid
Anti-inflammatory steroid
Inhaled
Butorphanol
Opioid
Analgesic
 receptor partial agonist
or antagonist
C3a, C5a
Inflammatory mediators
Anaphylatoxins
Low molecular weight complement
cleavage products
Calcium carbonate
Antiulcer
Antacid
Candesartan
Antihypertensive
Angiotensin receptor blocker
(ARB)
Captopril
Antihypertensive
Converting enzyme inhibitor
Heart failure treatment
Angioedema producer
Carbamazepine
Tricylic antidepressant (TCA)
Anticonvulsant
Carbenicillin
Penicillin antibiotic
Cell wall synthesis inhibitor
Antiulcer
Anti-pseudomonal penicillin
Inhibits peptidoglycan cross-linking
Carbidopa
Antiparkinson
Peripheral dopa decarboxylase
inhibitor
Carboprost
Oxytocic prostaglandin
Uterine stimulant
Carmustine (BCNU)
Antineoplastic
Alkylating Agent
Carteolol
Sympatholytic
 adrenergic antagonist
Antihypertensive
Bronchoconstrictor
Carvedilol
Sympatholytic
 adrenergic antagonist
Treatment for heart failure
Cascara
Contact cathartic
Anthraquinone derivative
Caspofungin
Echinocandin antifungal
Blocks synthesis of fungal
 (1,3)-d-glucan in the cell wall
Castor Oil
Contact cathartic
Cefaclor
Cephalosporin antibiotic
Cell wall synthesis inhibitor
2nd generation
Oral
Cefadroxil
Cephalosporin antibiotic
Cell wall synthesis inhibitor
1st generation
Oral
Cefepime
Cephalosporin antibiotic
Cell wall synthesis inhibitor
4th generation
CSF penetration
Cefotaxime
Cephalosporin antibiotic
Cell wall synthesis inhibitor
3rd generation
CSF penetration
Cefoxitin
Cephalosporin antibiotic
Cell wall synthesis inhibitor
2nd generation
Ceftazidime
Cephalosporin antibiotic
Cell wall synthesis inhibitor
3rd generation
Ceftriaxone
Cephalosporin antibiotic
Cell wall synthesis inhibitor
3rd generation
CSF penetration
Cefuroxime
Cephalosporin antibiotic
Cell wall synthesis inhibitor
2nd generation
CSF penetration
Celecoxib
NSAID
Anti-inflammatory
Cyclooxygenase 2 (COX-2) inhibitor
Cephalexin
Cephalosporin antibiotic
Cell wall synthesis inhibitor
1st generation
Oral
Cephalosporins
Antibiotics
 lactam
Cell wall synthesis inhibitors
Inhibit cross-linking of peptidoglycan
Cephalothin
Cephalosporin antibiotic
Cell wall synthesis inhibitor
1st generation
Oral
Cetirizine
Antihistamine
H1 antagonist
Non-sedating
Cetrorelix
Gonadotropin releasing hormone
antagonist
Synthetic GnRH analogue
Chloral hydrate
Sedative/Hypnotic
General anaesthetic
Barbiturate
Chloramphenicol
Antibiotic
Bacteriostatic protein synthesis inhibitor
50S ribosome
Inhibits peptide bond formation
Chlordiazepoxide
Sedative/hypnotic
Anxiolytic
Benodiazepine
Chloroquine
Antimalarial
Intercalates in DNA
Binds to ferriprotoporphyrin
Chlorpheniramine
Classical antihistamine
H1 antagonist
Chlorpromazine
Antipsychotic
Phenothiazine
Chlorpropamide
Oral hypoglycemic
Sulfonylurea
Insulinotropic
Chlorthalidone
Diuretic
Antihypertensive
Chlorothiazide
Thiazide diuretic
Na-Cl symporter inhibitor
Cholestyramine
Antihyperlipidemic
Bile acid binding resin (BABR)
Chorionic Gonadotropin
(hCG)
Gonadotropin
Ovulation inducing agent
Cidofovir
Antiherpes
Pyrimidine analog
Phosphorylated to inhibitor of viral
DNA polymerase
Cimetidine
Antihistamine
Antiulcer
H2 receptor antagonist
Ciprofloxacin
Fluoroquinolone antibiotic
DNA replication inhibitor
Inhibits bacterial DNA gyrase
Cisapride
Prokinetic agent
5HT4 agonist
Cisplatin
Antineoplastic
Miscellaneous
Cross-linking agent
Clarithromycin
Macrolide antibiotic
Bacteriostatic protein synthesis inhibitor
Antiulcer
50S ribosome
Inhibits translocation
Bacteriostatic
Clavulanic acid
-lactamase inhibitor
Combined with antibacterials
Clindamycin
Antibiotic
Bacteriostatic protein synthesis inhibitor
50S ribosome
Anaerobic infections
Clomiphene
Ovulation inducing agent
Partial estrogen agonist
Clonidine
Sympatholytic
2 adrenergic agonist
Antihypertensive
Clotrimazole
Imidazole antifungal
Inhibits synthesis of ergosterol
Lanosterol 14 demethylase inhibitor
Cloxacillin
Penicillin antibiotic
Cell wall synthesis inhibitor
Antiulcer
Penicillinase resistant penicillin
Inhibits peptidoglycan cross-linking
Clozapine
Antipsychotic
Clofibrate
Antihyperlipidemic
Lipoprotein lipase activator
Cobalamin
(cyanocobalamin, hydroxocobalamin)
Vitamin
Treatment for
vitamin B12 deficiency
Cocaine
Indirect sympathomimetic
Drug of abuse
Topical anaesthetic
Stimulant
Codeine
Opioid
Analgesic
Weak agonist
Colchicine
Antigout only
Anti-inflammatory
Microtubule inhibitor
Colestipol
Antihyperlipidemic
Bile acid binding resin (BABR)
Conjugated estrogens
Hormone
Estrogen
Used for HRT
Corticosterone
Adrenocorticosteroid
Glucosteroid
Cortisol (Hydrocortisone)
Adrenocorticosteroid
Glucocorticoid
Anti-inflammatory steroid
Corticotropin-releasing
Hormone (CRH)
Hypothalamic hormone
Stimulates release of ACTH
and -endorphin from the anterior
pituitary
Cromolyn sodium
Mast cell stabilizer
Inhibits release of
mast cell mediators
Used prophylactically in asthma
Cyclobenzaprine
Skeletal muscle relaxant
Cyclophosphamide
Antineoplastic
Alkylating Agent
Cycloserine
Antibiotic
Cell wall synthesis inhibitor
Secondary TB drug
Inhibits formation of Park nucleotide
Cyclosporine
Immunosuppressive
Antineoplastic
Binds cyclophilin
Inhibits calcineurin
Cyproterone acetate
Antiandrogen
Antineoplastic
Antrogen receptor antagonist
Cytarabine (AraC)
Antineoplastic
Antimetabolite
Dacarbazine
Antineoplastic
Alkylating Agent
Daclizumab
Immunosuppressive
Anti-CD25 (interleukin 2 receptor)
antibody
Organ transplant (anti-rejection)
Dactinomycin
Antineoplastic
Natural product
Antibiotic
Dalteparin
Anticoagulant
LMW Heparin
ATIII activator
Danthron
Contact cathartic
Anthraquinone derivative
Dantrolene
Skeletal muscle relaxant
Ryanodine receptor antagonist
Treatment for malignant hyperthermia
Dapsone
Sulfone antibiotic
Nucleic acid and
protein synthesis inhibitor
Inhibits dihydropteroate synthetase
Leprosy
Daunorubicin
Antineoplastic
Anthracycline antibiotic
Natural product
Deferoxamine
Antidote
Chelating agent
Removes iron
Delavirdine
Antiretroviral
Non-nucleoside reverse transcriptase
inhibitor (NNRTI)
Deprenyl/selegiline
Antiparkinson
Monoamine oxidase B inhibitor
(MAO-I)
Potentiates effects of L-Dopa
Desipramine
Tricyclic antidepressant (TCA)
Desmopressin acetate
(arginine vasopressin)
Antidiuretic hormone analogue
Plasma fraction used in treatment of
bleeding disorders
Desogesterel
Hormone
Progestin
19-nor testosterone analogue
Combination oral contraceptive
Dexamethasone
Adrenocorticosteroid
Glucocorticoid
Antineoplastic
Anti-inflammatory steroid
Not by inhalation
Dextromethorphan
Opioid
Antitussive
Diazepam
Sedative/hypnotic
Anxiolytic
Anticonvulsant
Benzodiazepine
Diazoxide
Vasodilator
Antihypertensive
Didanosine
Antiretroviral
Nucleoside reverse transcriptase
inhibitor (NRTI)
Dideoxyinosine (ddI)
Diethylcarbamazine
Antihelminthic
Treatment of intestinal
and tissue roundworms
Diethylstilbestrol
Hormone
Nonsteroidal estrogen
Diflunisal
NSAID
Analgesic, Anti-inflammatory
Antipyretic
Cyclooxygenase inhibitor
Digitalis
Cardiac glycoside
Antiarrhythmic
Na+/K+ ATPase inhibitor
Positive inotrope
Miscellaneous
(does not fit class I-IV organization)
Digitoxin
Cardiac glycoside
Antiarrhythmic
Na+/K+ ATPase inhibitor
Positive inotrope
Miscellaneous
(does not fit class I-IV organization)
Digoxin
Cardiac glycoside
Antiarrhythmic
Na+/K+ ATPase inhibitor
Positive inotrope
Miscellaneous
(does not fit class I-IV organization)
DIG-specific antibody
fragments
Antidote
Cardiac glycoside poisoning
Dihydrotestosterone
Hormone
Androgen
Natural male gonadal steroid
Diltiazem
Class IV antiarrhythmic
Antihypertensive
Ca2+ channel blocker
Dimenhydrinate
Antihistamine
Antiemetic
H1 receptor antagonist
Dinoprostone
(Dinoprost; PGE2)
Oxytocic prostaglandin
Uterine stimulant
Cervical ripener
Diphenhydramine
Classical antihistamine
Antiemetic
H1 antagonist
Diphenoxylate docusate
Antidiarrheal
Opiate
Dipyridamole
Antiplatelet
Phosphodiesterase inhibitor
(increases cAMP)
Disopyramide
Class I antiarrhythmic
Na+ channel blocker
(activated channels)
Dobutamine
Sympathomimetic
1 adrenergic agonist
Inotrope
Docusates
Lubricating laxatives
Stool softeners
Dofetilide
Class III antiarrhythmic
K+ channel blocker
Dopamine
Sympathomimetic
Inotrope
Vasodilator
Doxazosin
Sympatholytic
1 adrenergic antagonist
Antihypertensive
Doxorubicin
Antineoplastic
Anthracycline antibiotic
Natural product
Doxycycline
Tetracycline antibiotic
Bacteriostatic protein synthesis inhibitor
Antiulcer
30S ribosome
Prevents aminoacyl tRNA attachment
Dronabinol
Antiemetic
Cannabinoid
Drotrecogin alfa
(Activated Protein C)
Anticoagulant
Many actions
Treatment for septic shock
Dutasteride
Antiandrogen
Androgen synthesis inhibitor
5-reductase inhibitor
Echinacea purpurea
Dietary supplement
Immune system stimulant
Ecothiophate
Anticholinesterase
Vasodilator
Bronchoconstrictor
Glaucoma treatment
Edrophonium
Anticholinesterase
Vasodilator
Diagnostic for myaesthenia gravis
Bronchoconstrictor
Enalapril
Antihypertensive
Converting enzyme inhibitor
Angioedema producer
Enflurane
General anaesthetic
Inhaled anaesthetic
Enoxaparin
Anticoagulant
LMW Heparin
ATIII activator
Entacapone
Antiparkinson
Catechol-o-methyltransferase
inhibitor
Ephedra
(Ma Huang)
Dietary supplement
Amphetamine-like stimulant
Ephedrine
Indirect sympathomimetic
Vasoconstrictor
Bronchodilator
Decongestant
Epinephrine
Sympathomimetic
 and  adrenergic agonist
Vasoconstrictor
Bronchodilator
Eprosartan
Antihypertensive
Angiotensin receptor blocker
(ARB)
Ergonovine
Oxytocic ergot alkaloid
Uterine stimulant
Erythromycin
Macrolide antibiotic
Bacteriostatic protein synthesis inhibitor
Antiulcer
50S ribosome
Inhibits translocation
Erythropoietin (EPO)
Cytokine
Primary regulator of RBC synthesis
Esmolol
Sympatholytic
1 adrenergic antagonist
Class II Antiarrythmic
Antihypertensive
Bronchoconstrictor
Estraderm
Hormone
Estrogen
Transdermal formulation
Estradiol
Hormone
Estrogen
Primary natural female gonadal
steroid
Estriol
Hormone
Estrogen
Natural female gonadal steroid
Estrone
Hormone
Estrogen
Natural female gonadal steroid
Etanercept
TNF inhibitor
Tumor necrosis factor receptor
+ Fc portion of IgG
Used in rheumatoid arthritis
Ethacrynic acid
Loop diuretic
Na-K-2Cl symporter inhibitor
Ethambutol
Antibiotic
Major drug for tuberculosis
Ethanol
Drug of abuse
Sedative
Ethinyl estradiol
Hormone
Estrogen
Synthetic femal gonadal steroid
Combination oral contraceptive
Ethionamide
Antibiotic
Secondary drug for tuberculosis
Etidronate
Anti-osteoporesis
Bisphosphonate
Inhibitor of osteoclast-mediated
bone resorption
Etoposide
Antineoplastic
Natural product
Plant alkaloid
Ethosuximide
Anticonvulsant
Etomidate
General anaesthetic
Intravenous anaesthetic
Exemestane
Antineoplastic
Antiestrogen
Aromatase Inhibitor
Ezitimibe
Antihyperlipidemic
Cholesterol absorption inhibitor
Famciclovir
Antiherpes
Purine analog
Phosphorylated to an inhibitor of
viral DNA polymerase
Famotidine
Antihistamine
Antiulcer
H2 receptor antagonist
Felodipine
Antihypertensive
Calcium channel blocker
Fenofibrate
Antihyperlipidemic
Lipoprotein lipase activator
Fentanyl
Opioid
Analgesic
 receptor agonist
Fexofenadine
Antihistamine
H1 antagonist
Non-sedating
Finasteride
Antiandrogen
Androgen synthesis inhibitor
5-reductase inhibitor
Flecainide
Class I antiarrhythmic
Na+ channel blocker
Fluconazole
Triazole antifungal
Inhibits synthesis of ergosterol by
inhibiting lanosterol 14 demethylase
Flucytosine
Antifungal
Converted by fungi to 5-fluorouracil
 faulty RNA and DNA synthesis
Fludrocortisone
Adrenocorticosteroid
Mineralocorticoid
Flumazenil
Benzodiazepine antagonist
Flunisolide
Adrenocorticosteroid
Glucocorticoid
Anti-inflammatory steroid
Inhaled
Fluorinated Quinolones
ciprofloxacin, norfloxacin
Antibiotics
DNA replication inhibitors
Inhibit bacterial DNA gyrase
5-Fluorouracil
Antineoplastic
Antimetabolite
Thymidylate synthase inhibitor
Fluoxetine
Antidepressant
Selective serotonin reuptake inhibitor
(SSRI)
Flurazepam
Sedative/Hypnotic
Benzodiazepine
Flutamide
Antiandrogen
Antineoplastic
Antrogen receptor antagonist
Fluticasone
Adrenocorticosteroid
Glucocorticoid
Anti-inflammatory steroid
Inhaled
Fluvastatin
Antihyperlipidemic
HMG-CoA Reductase Inhibitor
Folic acid
Vitamin
Treatment for folic
acid deficiency
Follicle-Stimulating Hormone
(FSH)
Anterior pituitary hormone
Regulator of gonadal function
Formoterol
Sympathomimetic
2 adrenergic agonist
Long acting bronchodilator
Foscarnet
Antiherpes
Pyrophosphate analog
Directly inhibits viral DNA
polymerase
Fosinopril
Antihypertensive
Converting enzyme inhibitor
Fulvestrant
Antineoplastic
Antiestrogen
Estrogen receptor antagonist
Furosemide
Loop diuretic
Na-K-2Cl symporter inhibitor
Antihypertensive
Ganciclovir
Antiherpes
Purine analog
Phosphorylated to an inhibitor
of viral DNA polymerase
Ganirelix
Gonadotropin releasing hormone
antagonist
Synthetic GnRH analogue
Gemfibrozil
Antihyperlipidemic
Lipoprotein lipase activator
Gemtuzumab
Antineoplastic
Anti-CD33 antibody
Gentamicin
Aminoglycoside antibiotic
Bactericical protein synthesis inhibitor
30S ribosome
Freezes initiation
Ginko biloba
Dietary supplement
Treatment of Alzheimer symptoms
Ginko biloba
Dietary supplement
Improvement in energy and vitality
Glargine insulin
Hormone
Insulin analogue
Long acting
Glimepiride
Oral hypoglycemic
Sulfonylurea
Insulinotropic
Glipizide
Oral hypoglycemic
Sulfonylurea
Insulinotropic
Glutethimide
Sedative/Hypnotic
Glyburide
Oral hypoglycemic
Sulfonylurea
Insulinotropic
Gold salts
auranofin, aurothioglucose
Disease modifying anti-rheumatic
drugs (DMARD)
Gonadorelin
Gonadotropin releasing hormone
(GnRH)
Sulfonylurea
Insulinotropic
Gonadotropin-releasing
Hormone (GnRH)
Hypothalamic hormone
Stimulates release of FSH and LH
from the anterior pituitary
Goserelin
Antineoplastic
Gonadotropin releasing hormone
(GnRH) analogue
Granulocyte-Colony
Stimulating Factor (G-CSF)
Cytokine
Granulocytes synthesis stimulator
Granulocyte/Monocyte-Colony
Stimulating Factor (GM-CSF)
Cytokine
WBC (granulocytes and monocyte)
synthesis stimulator
Griseofulvin
Antifungal
Binds to microtubules
Growth Hormone-releasing
Hormone (GHRH)
Hypothalamic hormone
Stimulates release of growth hormone
from the anterior pituitary
Growth Hormone
Somatotropin
(GH)
Anterior pituitary hormone
Stimulates insulin-like growth factor
I release ( growth at open epiphyses),
lipolysis and skeletal muscle growth
Guanabenz
Sympatholytic
Antihypertensive
Guanadrel
Sympatholytic
Antihypertensive
Guanethidine
Sympatholytic
Antihypertensive
Guanfacine
Sympatholytic
2 adrenergic agonist
Antihypertensive
Haloperidol
Antipsychotic
Halothane
General anaesthetic
Inhaled anaesthetic
Heparin
Anticoagulant
ATIII activator
Heroin
Drug of abuse
Opioid
Hirudin
Anticoagulant
Thrombin inhibitor
Histamine
Inflammatory mediator
Stored in mast cells and basophils
Histrelin
Gonadotropin releasing hormone
(GnRH) agonist
Synthetic GnRH analogue
Human Chorionic Gonadotropin
(HCG)
Placental hormone
Stimulates ovarian
progesterone production
Maintains placenta
Hydralazine
Vasodilator
Antihypertensive
Hydrochlorothiazide
Thiazide diuretic
Na-Cl symporter inhibitor
Antihypertensive
Hydrocortisone
Adrenocorticosteroid
Glucocorticoid
Anti-inflammatory steroid
Hydroxychloroquine
Disease modifying
anti-rheumatic drug (DMARD)
4-Hydroxycoumarin
Oral anticoagulant
Vitamin K synthesis inhibitor
Hydroxyurea
Antineoplastic
Miscellaneous
Ribonucleotide reductase inhibitor
Hydroxyzine
Classical antihistamine
H1 antagonist
Ibritumomab
Antineoplastic
Anti-CD20 antibody
Ibuprofen
NSAID
Analgesic, Anti-inflammatory
Antipyretic
Irreversible cyclooxygenase inhibitor
Ibutilide
Class III antiarrhythmic
K+ channel blocker
Imatinib
Antineoplastic
Miscellaneous
Tyrosine kinase inhibitor
Imipenem
New  lactam antibiotic
Carbapenem, combined with cilastatin
which inhibits a dipeptidase that
inactivates imipenem
Imipramine
Indirect sympathomimetic
Tricyclic antidepressant (TCA)
Antimicturant
Indapamide
Thiazide-like diuretic
Na-Cl symporter inhibitor
Antihypertensive
Indinavir
Antiretroviral
Protease inhibitor (PI)
Indomethacin
NSAID
Analgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
Tocolytic
Uterine relaxant
Infliximab
TNF inhibitor
Anti-TNF monoclonal antibody
Insulin
Hormone
Insulin analogue
Short acting
Interferon alpha
Antiviral for hepatitis
Antineoplastic
Cytokine
Anti-angiogenesis
Interleukin 2
Cytokine
Antineoplastic
Interleukin 11
Cytokine
Antineoplastic (supporting agent)
Iodide
Antithyroid
Prevents synthesis and release of
thyroid hormones
(blocks iodine organification)
Decreases hyperplasia
Iodoquinol
Antiparasitic
Treatment of protozoal infections
Ipecac
Emetic
Ipratropium
Anticholinergic
Antimuscarinic
Inhaled
Bronchodilator
Irbesartan
Antihypertensive
Angiotensin receptor blocker
(ARB)
Iressa
Antineoplastic
Miscellaneous
Tyrosine kinase inhibitor
Iron
(ferrous sulfate, iron dextran)
Essential nutrient
Required for hemoglobin and
myoglobin synthesis
Isoetharine
Sympathomimetic
 adrenergic agonist
Bronchodilator
Isoflurane
General anaesthetic
Inhaled anaesthetic
Isoniazid
Antibiotic
Inhibits biosynthesis of mycolic acids
Major drug for tuberculosis
Isoproterenol
Sympathomimetic
 adrenergic agonist
Vasodilator
Bronchodilator
Isosorbide dinitrate
Venodilator
Used to treat CHF
Isradipine
Antihypertensive
Calcium channel blocker
Itraconazole
Triazole antifungal
Inhibits synthesis of ergosterol by
inhibiting lanosterol 14 demethylase
Ivermectin
Antihelminthic
Treatment of intestinal
and tissue roundworms
Kallidin
Inflammatory mediator
Plasma, hypotension, pain
Kava kava
Dietary supplement
Stress relief and
treatment of insomnia
Ketamine
General anaesthetic
Drug of abuse
Sedative
Ketoconazole
Imidazole antifungal
Inhibits synthesis of ergosterol by
inhibiting lanosterol 14 demethylase
Ketoprofen
NSAID
Analgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
Labetalol
Sympatholytic
 and  adrenergic antagonist
Antihypertensive
Lactulose
Saline (osmotic) cathartic
Lamivudine
Antiretroviral
Nucleoside reverse transcriptase
inhibitor (NRTI)
Lente insulin
Hormone
Insulin analogue
Intermediate acting
Lepirudin
Anticoagulant
Thrombin inhibitor
Letrozole
Antineoplastic
Antiestrogen
Aromatase Inhibitor
Leukotriene B4 (LTB4)
Inflammatory mediator
Lipoxygenase product
of arachidonate metabolism
Chemotactic
Leukotrienes C4, D4, E4
(LTC4, LTD4, LTE4)
Inflammatory mediators
Cysteinyl leukotrienes
Peptidyl leukotrienes
SRS-A
Lipoxygenase products of
arachidonate metabolism
Leucovorin
Antineoplastic (supporting agent)
Folic acid analogue
(used in methotrexate rescue)
Leuprolide
Antineoplastic
Gonadotropin releasing hormone
(GnRH) analogue
Levobunolol
Sympatholytic
 adrenergic antagonist
Antihypertensive
Bronchoconstrictor
Levodopa
Antiparkinson
Dopamine agonist
Inhibits growth hormone release
Levonorgestrel
Hormone
Progestin
19-nor testosterone analogue
Combination oral contraceptive
Levothyroxine (T4)
Thyroid hormone
Lidocaine
Class I antiarrhythmic
Local anaesthetic
Na+ channel blocker
(activated and inactivated channels)
Linezolid
Oxazolidinone antibiotic
Protein synthesis inhibitor
50S ribosomal subunit
Liothyronine (T3)
Thyroid hormone
Lisinopril
Antihypertensive
Converting enzyme inhibitor
Heart failure treatment
Angioedema producer
Lispro insulin
Hormone
Insulin analogue
Ultra short acting
Lithium
Antidepressant
Used to treat
manic/depressive disorder
Lomustine (CCNU)
Antineoplastic
Alkylating Agent
Loperamide
Antidiarrheal
Opiate
Loratidine
Antihistamine
H1 antagonist
Non-sedating
Lorazepam
Anxiolytic
Anticonvulsant
Losartan
Antihypertensive
Angiotensin receptor blocker
(ARB)
Lovastatin
Antihyperlipidemic
HMG-CoA Reductase Inhibitor
Lutenizing Hormone (LH)
Anterior pituitary hormone
Regulator of gonadal function
Lypressin
Antidiuretic hormone analogue
Lysergic acid diethylamide
(LSD)
Drug of abuse
Hallucinogen
Macrolides
erythromycin, azithromycin, clarithromycin
Antibiotics
Bacteriostatic protein synthesis inhibitors
50S ribosome
Magnesium hydroxide
Antiulcer
Saline (osmotic) cathartic
Antacid
Magnesium sulfate
Calcium antagonist
Tocolytic
Uterine relaxant
Malathion
Anticholinesterase
Vasodilator
Bronchoconstrictor
Mannitol
Osmotic diuretic
Marijuana
Drug of abuse
Cannabinoid
Mebendazole
Antihelminthic
Treatment of intestinal roundworms
Meclizine
Antihistamine
Antiemetic
H1 receptor antagonist
Meclofenamate
NSAID
Analgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
Mechlorethamine
Antineoplastic
Alkylating Agent
Medroxyprogesterone
Hormone
Progestin
Synthetic progesterone analogue
Contraceptive
Mefloquine
Antimalarial
Treatment and prophylaxis for
chloroquine resistant Plasmodium
Meglumine antimonate
Tropical antiparasitic
Organic antimonial
Treatment of Leishmaniasis
Melarsoprol
Tropical antiparasitic
Treatment of African
Trypanosomiasis in CNS
Melphalan
Antineoplastic
Alkylating Agent
Menotropin
Gonadotropin
Ovulation inducing agent
Meperidine
Opioid analgesic
 receptor agonist
Mepivacaine
Local anaesthetic
Meprobamate
Sedative/hypnotic
Anxiolytic
6-Mercaptopurine
Antineoplastic
Antimetabolite
(“pseudofeedback inhibition” of
HGPRT and PRP – purine synthesis)
Mesalamine
(5-ASA)
NSAID (salicylate)
Mesna
Antineoplastic (supporting agent)
Prevent hemorrhagic cystitis
due to cyclophosphamide
Mestranol
Hormone
Estrogen
Synthetic female gonadal steroid
Combination oral contraceptive
Metalazone
Diuretic
Antihypertensive
Metamphetamine
Drug of abuse
Stimulant
Metaproterenol
Sympathomimetic
2 adrenergic agonist
Bronchodilator
Used in asthma
Metformin
Oral hypoglycemic
Biguanide
Hepatic gluconeogenesis inhibitor
Methacholine
Cholinomimetic
Bronchoconstrictor
Methadone
Opioid
 receptor agonist
Methenamine
Urinary tract antiseptic
Decomposes to formaldehyde
in acidic environment
Methicillin
Penicillin antibiotic
Cell wall synthesis inhibitor
Pencillinase resistant penicillin
Inhibits peptidoglycan cross-linking
Methimazol
Antithyroid
Prevents synthesis of
thyroid hormones
(blocks iodine organification)
Methotrexate
Immunosuppressive
Antineoplastic
Folic acid antagonist
Dihydrofolate reductase inhibitor
Methoxamine
Sympathomimetic
1 adrenergic agonist
Vasoconstrictor
Methylcellulose
Bulk laxative
Methydopa
Sympatholytic
2 adrenergic agonist
Antihypertensive
Methylphenidate
Indirect sympathomimetic
Drug of abuse
ADD treatment
Stimulant
Methylprednisolone
Adrenocorticosteroid
Glucocorticoid
Anti-inflammatory steroid
Not by inhalation
Methyltestosterone
Hormone
Androgen
Synthetic oral
Metipranolol
Sympatholytic
 adrenergic antagonist
Bronchoconstrictor
Metoclopramide
Prokinetic agent
Antiemetic
D2 antagonist
Metocurine
Paralytic
Paralyzes skeletal muscles
Metolazone
Thiazide-like diuretic
Na-Cl symporter inhibitor
Metoprolol
Sympatholytic
1 adrenergic antagonist
Antihypertensive
Heart failure medication
Bronchoconstrictor
Metronidazole
Antibiotic
Antiparasitic
Antiulcer
Anaerobes
Reduction leads to intermediates
that damage DNA
Metyrapone
Glucocorticoid antagonist
Mexilitine
Class I antiarrhythmic
Na+ channel blocker
(activated and inactivated channels)
Miconazole
Imidazole antifungal
Inhibits synthesis of ergosterol by
inhibiting lanosterol 14 demethylase
Midazolam
Sedative hypnotic
Short-acting benzodiazopine
Mifepristone
(RU-486)
Progesterone antagonist
Miglitol
Oral hypoglycemic
Alpha-glucosidase inhibitor
Inhibits intestinal glucose absorption
Mineral oil
Lubricating laxative
Stool softener
Minocycline
Tetracycline Antibiotic
Bacteriostatic protein synthesis inhibitor
Antiulcer
30S ribosome
Prevents aminoacyl tRNA attachment
Minoxidil
Vasodilator
Antihypertensive
Misoprostol
Prostaglandin
Mitomycin C
Antineoplastic
Natural product
Antibiotic
Mivacurium
Paralytic
Paralyzes skeletal muscles
Moezipril
Antihypertensive
Converting enzyme inhibitor
Montelukast
Leukotriene inhibitor
LTR1 and LTD4 antagonist
Asthma treatment
Moricizine
Class I antiarrhythmic
Na+ channel blocker
Morphine
Opioid
Analgesic
 receptor agonist
Muromonab-CD3
Immunosuppressive
Mouse monoclonal anti-CD3 antibody
Organ transplant (anti-rejection)
Mycophenolate
Immunosuppressive
Inhibits inosine monophosphate
dehydrogenase activity
Nadolol
Sympatholytic
 adrenergic antagonist
Antihypertensive
Nafarelin
Gonadotropin releasing hormone
(GnRH) agonist
Nafcillin
Penicillin antibiotic
Cell wall synthesis inhibitor
Antiulcer
Penicillinase resistant penicillin
Inhibits peptidoglycan cross-linking
Nalbuphine
Opioid antagonist
 receptor antagonist
Nalidixic acid
Urinary tract antiseptic
Quinolone
Inhibits bacterial DNA gyrase
Nalmefene
Opioid antagonist
Nalorphine
Opioid antagonist
Naloxone
Opioid antagonist
Naproxen
NSAID
Analgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
Nateglinide
Oral hypoglycemic
Meglitinide
Insulinotropic
Naltrexone
Opioid antagonist
Nedocromil
Mast cell stabilizer
Inhibits release of mast cell
mediators
Used prophylactically in asthma
Neomycin
Aminoglycoside antibiotic
Bactericidal protein synthesis inhibitor
30S ribosome
Freezes initiation
Topical
Neostigmine
Anticholinesterase
Vasodilator
Treatment for myaesthenia gravis
Promotes defecation and urination
Bronchoconstrictor
Netilmicin
Aminoglycoside antibiotic
Bactericidal protein synthesis inhibitor
30S ribosome
Freezes initiation
Nevirapine
Antiretroviral
Non-nucleoside reverse transcriptase
inhibitor (NNRTI)
Nicardipine
Antihypertensive
Calcium channel blocker
Nicotine
Cholinomimetic
Drug of abuse
Nicotinic receptor agonist
(skeletal muscle contraction)
Stimulant
Smoking cessation medication
Nicotinic acid
Antihyperlipidemic
Inhibition of VLDL secretion (?)
Nifedipine
Antihypertensive
Antianginal
Calcium channel blocker
Nifurtimox
Tropical antiparasitic
Treatment of South American
Trypanosomiasis; Chagas disease
Nisoldipine
Antihypertensive
Calcium channel blocker
Nitrendipine
Antihypertensive
Calcium channel blocker
Nitrofurantoin
Urinary tract antiseptic
Reduction leads to intermediates that
damage DNA
Nitroglycerine
Venodilator
Antianginal
Nitroprusside
Vasodilator
Antihypertensive
Nitrous oxide
General anaesthetic
Inhaled anaesthetic
Nizatidine
Antihistamine
Antiulcer
H2 receptor antagonist
Norepinephrine
Sympathomimetic
Vasoconstrictor
Norethindrone
Hormone
Progestin
19-nor testosterone analogue
Combination oral contraceptive
Norethynodrel
Hormone
Progestin
19-nor testosterone analogue
Combination oral contraceptive
Norfloxacin
Fluoroquinolone antibiotic
DNA replication inhibitor
Inhibits bacterial DNA gyrase
Norgestimate
Hormone
Progestin
19-nor testosterone analogue
Combination oral contraceptive
Norgestrel
Hormone
Progestin
19-nor testosterone analogue
Combination oral contraceptive
Nortriptyline
Tricyclic antidepressant (TCA)
NPH insulin
Hormone
Insulin analogue
Intermediate acting
Non-steroidal
Anti-inflammatory Drugs
(NSAIDs)
Analgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitors
Nystatin
Antifungal
Polyene antibiotic
Binds to ergosterol & alters permeability
Topical
Octreotide
Somatostatin analogue
Peptide hormone inhibitor
Decreases growth hormone secretion
Decreases gastric and pancreatic
secretions
Ondansetron
Antiemetic
5HT3 receptor antagonist
Olsalazine
NSAID (salicylate)
Omeprazole
Antiulcer
H+/K+ ATPase inhibitor
Organic antimonials
sodium stibogluconate
meglumine antimonate
Tropical antiparasitic
Treatment of Leishmaniasis
Oseltamivir
Antiviral
Inhibits neuraminidase and
decreases viral release
Treatment of Influenza A & B
Oxacillin
Penicillin antibiotic
Cell wall synthesis inhibitor
Antiulcer
Pencillinase resistant penicillin
Inhibits peptidoglycan cross-linking
Oxazepam
Sedative/hypnotic
Anxiolytic
Benzodiazepine
Oxybutinin
Anticholinergic
Muscarinic receptor antagonist
Prevents urination
Oxycodone
Analgesic
Opioid agonist
Oxytetracycline
Tetracycline antibiotic
Bacteriostatic protein synthesis inhibitor
Antiulcer
30S ribosome
Prevents aminoacyl tRNA attachment
Oxytocin
Hypothalamic (posterior pituitary)
hormone
Uterine stimulant
Paclitaxel
Antineoplastic
Natural product
Plant alkaloid (taxane)
Palivizumab
Antiviral
Monoclonal antibody against
the surface of
respiratory syncytial virus
Pamidronate
Anti-osteoporesis
Bisphosphonate
Inhibitor of osteoclast-mediated
bone resorption
Pancuronium
Paralytic
Paralyzes skeletal muscles
Pantoprazole
Antiulcer
H+/K+ ATPase inhibitor
Para-aminosalicylic acid
Antibiotic
Nucleic acid and
protein synthesis inhibitor
Inhibits dihydropteroate synthetase
Secondary TB drug
Paraldehyde
Sedative/Hypnotic
Parathyroid hormone
Hormone
Maintains plasma Ca2+ concentrations
Paromomycin
Antiparasitic
Aminoglycoside antibiotic
Treatment of protozoal infections
Penbutolol
Sympatholytic
 adrenergic antagonist
Antihypertensive
Bronchoconstrictor
Penciclovir
Antiherpes
Purine analog
Phosphorylated to inhibitor of viral
DNA polymerase
Penicillins
 lactam antibiotics
Cell wall synthesis inhibitors
Inhibit cross-linking of peptidoglycan
Penicillin G
Penicillin antibiotic
Cell wall synthesis inhibitor
Antiulcer
Acid labile
Inhibits peptidoglycan cross-linking
Penicillin V
Penicillin antibiotic
Cell wall synthesis inhibitor
Antiulcer
More acid resistant than Penicillin G
Inhibits peptidoglycan cross-linking
Pentamidine
Tropical antiparasitic
Treatment of African
Trypanosomiasis
Pentazocine
Opioid analgesic
 receptor partial agonist or
antagonist
Pentobarbital
Sedative/Hypnotic
Barbiturate
Pentostatin
Antineoplastic
Miscellaneous
Enzyme inhibitor
(blocks purine synthesis)
Perindopril
Antihypertensive
Converting enzyme inhibitor
Phencyclidine (PCP)
Drug of abuse
Hallucinogen
Phenobarbital
Sedative/Hypnotic
Anticonvulsant
Barbiturate
Phenoxybenzamine
Sympatholytic
 adrenergic antagonist
Antihypertensive
Phentolamine
Sympatholytic
 adrenergic antagonist
Antihypertensive
Phenylephrine
Sympathomimetic
1 adrenergic agonist
Vasoconstrictor
Nasal decongestant
Phenylpropanolamine
Indirect sympathomimetic
Nasal decongestant
Removed from market*
(may be in medicine cabinets!)
Phenytoin
Anticonvulsant
Class I antiarrhythmic
Na+ channel blocker
(inactivated channels)
Physostigmine
Anticholinesterase
Bradycardic
Vasodilator
Bronchoconstrictor
Phytonadione
Vitamin K
Warfarin antagonist
Pilocarpine
Cholinomimetic
Muscarinic agonist
Antiglaucoma
Bronchoconstrictor
Pindolol
Sympatholytic
 adrenergic antagonist
Antihypertensive
Bronchoconstrictor
Pioglitazone
Oral hypoglycemic
Thiazolidinedione
Insulin sensitizer
Pipecuronium
Paralytic
Paralyze skeletal muscles
Piperacillin
Penicillin antibiotic
Cell wall synthesis inhibitor
Antiulcer
Anti-pseudomonal penicillin
Inhibits peptidoglycan cross-linking
Pirbuterol
Sympathomimetic
2 adrenergic agonist
Bronchodilator
Piroxicam
NSAID
Analgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
Platelet Activating Factor
(PAF)
Inflammatory mediator
Lipid
Hypotensive
Polymyxin B
Antibiotic
Disrupts gram negative cell membrane
Binds phosphatidylethanolamine
Bactericidal
Pralidoxime
Antidote
Cholinesterase reactivator
Pramipexole
Antiparkinson
Dopamine agonist (non-ergot)
Pravastatin
Antihyperlipidemic
HMG-CoA Reductase Inhibitor
Prazosin
Sympatholytic
1 adrenergic antagonist
Antihypertensive
Praziquantel
Antihelminthic
Treatment of trematode (fluke) and
cestode (tapeworm) infections
Prednisone
Adrenocorticosteroid
Glucocorticoid
Antineoplastic
Anti-inflammatory
Not by inhalation
Primaquine
Antimalarial
Eliminates hepatic forms of
plasmodium
Primidone
Anticonvulsant
Probenecid
Uricosuric
Adjunct in penicillin therapy
Probucol
Antihyperlipidemic
LDL oxidation inhibitor
Procainamide
Class I antiarrhythmic
Na+ channel blocker
(activated channels)
Procaine
Local anaesthetic
Procaine Penicillin G
Penicillin antibiotic
Cell wall synthesis inhibitor
Repository preparation
Inhibits peptidoglycan cross-linking
Procarbazine
Antineoplastic
Miscellaneous
Probably acts as alkylating agent
Prochlorperazine
Antiemetic
D2 receptor antagonist
Phenothiazine
Progesterone
Hormone
Progestin
Natural female progestin
Proguanil
Antimalarial
Inhibits plasmodial dihydrofolate
reductase
Prolactin
Anterior pituitary hormone
Regulator of lactation
Promethazine
Classical antihistamine
Antipsychotic
Antiemetic
H1 antagonist
Propafenone
Class I antiarrhythmic
Na+ channel blocker
Weak -blocker
Propofol
General anaesthetic
Intravenous anaesthetic
Propranolol
Sympatholytic
 adrenergic antagonist
Class II antiarrythmic
Antihypertensive
Bronchoconstrictor
Propylthiouracil
Antithyroid
Prevents synthesis of
thyroid hormones
(blocks iodine organification)
Prostaglandin D2 (PGD2)
Bronchoconstrictor
Cyclooxygenase product of
arachidonate metabolism
Prostaglandin E2 (PGE2)
Inflammatory mediator
Cyclooxygenase product of
arachidonate metabolism
Prostaglandin F2 (PGF2)
Inflammatory mediator
Cyclooxygenase product of
arachidonate metabolism
Prostaglandin I2 (PGI2)
Prostacyclin
Inflammatory mediator
Inhibits platelet aggregation
Cyclooxygenase product of
arachidonate metabolism
Protamine Sulfate
Heparin antagonist
Pseudoephedrine
Sympathomimetic
 and  adrenergic agonist
Vasoconstrictor
Nasal decongestant
Psyllium hydrophilic
mucilloid
Bulk laxative
Pyrantel Pamoate
Antihelminthic
Treatment of intestinal roundworms
Pyrazinamide
Antibiotic
Major drug for tuberculosis
Pyridostigmine
Anticholinesterase
Vasodilator
Treatment for myaesthenia gravis
Bronchoconstrictor
Pyrimethamine
Antimalarial
Protein and nucleic acid synthesis
inhibitor
Plasmodial dihydrofolate reductase
inhibitor
Quinapril
Antihypertensive
Converting enzyme inhibitor
Quinethazone
Thiazide-like diuretic
Na-Cl symporter inhibitor
Quinidine
Antimalarial
Protein and nucleic acid
synthesis inhibitor
Class I antiarrhythmic
Intercalates in DNA
Binds to ferriprotoporphyrin
Na+ channel blocker
Quinine
Antimalarial
Intercalates in DNA
Binds to ferriprotoporphyrin
Quinopristin/Dalfopristin
Streptogramin antibiotic
Protein synthesis inhibitor
50S ribosomal subunit
Radioactive Iodide
131
( I)
Antithyroid
Destruction of thyroid parenchyma
Raloxifene
Antiestrogen
Selective estrogen receptor
modulator (SERM)
Ramipril
Antihypertensive
Converting enzyme inhibitor
Ranitidine
Antihistamine
Antiulcer
H2 receptor antagonist
Repaglinide
Oral hypoglycemic
Meglitinide
Insulinotropic
Reserpine
Sympatholytic
Antihypertensive
Resperidone
Antipsychotic
Reteplase
Thrombolytic
Tissue plasminogen activator (tPA)
Ribavirin
Antiviral
Primarily used as aerosol for
respiratory syncytial virus
Rifampin
Antibiotic
Nucleic acid synthesis inhibitor
Inhibits DNA dependent RNA polymerase
Major drug for TB
Rimantadine
Antiviral
Inhibits replication
at the stage of uncoating
Treatment of Influenza A
Ritodrine
Sympathomimetic
2 adrenergic agonist
Tocolytic
Uterine relaxant
Ritonavir
Antiretroviral
Protease inhibitor (PI)
Rituxumab
Antineoplastic
Anti-CD20 antibody
Rocuronium
Paralytic
Paralyzes skeletal muscles
Rofecoxib
NSAID
Anti-inflammatory
Cyclooxygenase 2 (COX-2) inhibitor
Ropinirole
Antiparkinson
Dopamine agonist (non-ergot)
Rosiglitazone
Oral hypoglycemic
Thiazolidinedione
Insulin sensitizer
Salmeterol
Sympathomimetic
2 adrenergic agonist
Long acting bronchodilator
Saquinavir
Antiretroviral
Protease inhibitor (PI)
Saw palmetto
Dietary supplement
Treatment for benign prostatic
hyperplasia (BPH)
Senna
Contact cathartic
Anthraquinone derivative
Scopolamine
Anticholinergic
Antiemetic
Muscarinic receptor antagonist
Sertraline
Antidepressant
Selective serotonin reuptake inhibitor
(SSRI)
Sildenafil
Vasodilator
Promotes erection
Silver sulfadiazine
Sulfonamide antibiotic
Microbial nucleic acid
and protein synthesis inhibitor
Inhibits dihydropteroate synthetase
Topical
Simethicone
Anti-flatulent
Simvastatin
Antihyperlipidemic
HMG-CoA Reductase Inhibitor
Sirolimus
Rapamycin
Immunosuppressive
Binds FKBP, inhibits mTOR
(mammalian kinase target of
rapamycin) & cell cycle progression
Sodium bicarbonate
Antiulcer
Antidote
Antacid
Alkalinization of urine to treat drug
toxicity (esp. barbiturates, salicylates, methanol)
Sodium phosphate
Saline (osmotic) cathartic
Sodium stibogluconate
Tropical antiparasitic
Organic antimonial
Treatment of Leishmaniasis
Somatostatin
Somatotropin Release-inhibiting Hormone
(SRIH)
Hypothalamic hormone
Inhibits release of growth hormone
from the anterior pituitary
Somatrem
Growth hormone analogue
Stimulates insulin-like growth factor
I release ( growth at open epiphyses),
lipolysis and skeletal muscle growth
Somatropin
Growth hormone analogue
Stimulates insulin-like growth factor
I release ( growth at open epiphyses),
lipolysis and skeletal muscle growth
Sotolol
Class II antiarrythmic
Sympatholytic
 adrenergic antagonist
Spectinomycin
Antibiotic
Bacteriostatic protein synthesis inhibitor
30S ribosome
Spironolactone
Potassium sparing diuretic
Antiandrogen
Aldosterone receptor antagonist
Androgen receptor antagonist
Testosterone synthesis inhibitor
Antihypertensive
Heart failure treatment
St. John’s Wort
Dietary supplement
Antidepressant
Streptokinase
Thrombolytic
Streptomycin
Aminoglycoside antibiotic
Bactericidal protein synthesis inhibitor
30S ribosome
Freezes initiation
Succinylcholine
Paralytic
Depolarizing blocker
Paralyzes skeletal muscles
Bronchoconstrictor
Sucralfate
Antiulcer
Sufentanil
Opioid
General anaesthetic
Intravenous anaesthetic
Sulfacetamide
Sulfonamide antibiotic
Microbial nucleic acid
and protein synthesis inhibitor
Inhibits dihydropteroate synthetase
Topical
Sulfadoxine
Sulfonamide antibiotic
Microbial nucleic acid
and protein synthesis inhibitor
Dihydropteroate synthetase inhibitor
Sulfamethoxazole
Sulfonamide antibiotic
Microbial nucleic acid
and protein synthesis inhibitor
Inhibits dihydropteroate synthetase
Sulfasalazine
Disease modifying
anti-rheumatic drug (DMARD)
Metabolized to sulfonamide
+ salicylate (NSAID)
Sulfinpyrazone
Uricosuric
Anti-gout
Sulfisoxazole
Sulfonamide antibiotic
Nucleic acid and
protein synthesis inhibitor
Inhibits dihydropteroate synthetase
Sulfonamides
Antibiotics
Nucleic acid and
protein synthesis inhibitors
Inhibit dihydropteroate synthetase
Sulindac
NSAID
Analgesic, Anti-inflammatory,
Antipyretic
Cyclooxygenase inhibitor
Suramin
Tropical antiparasitic
Treatment of African
Trypanosomiasis
Tacrolimus
Immunosuppressive
Antineoplastic
Binds FKBP (FK506 binding protein)
Inhibits calcineurin
Tamoxifen
Antineoplastic
Antiestrogen
Estrogen receptor anatagonist
Telmisartan
Antihypertensive
Angiotensin receptor blocker
(ARB)
Temazepam
Sedative/Hypnotic
Benzodiazepine
Tenecteplase
Thrombolytic
Tissue plasminogen activator (tPA)
Terazosin
Sympatholytic
1 adrenergic antagonist
Antihypertensive
Treatment for benign prostatic
hypertrophy
Terbinafine
Allylamine antifungal
Inhibits ergosterol synthesis by
inhibiting squalene epoxidase
Terbutaline
Sympathomimetic
2 adrenergic agonist
Short acting bronchodilator
Tocolytic
Uterine relaxant
Testosterone
Hormone
Androgen
Natural male gonadal steroid
Testosterone cypionate
Hormone
Androgen
Synthetic depot
Testosterone enanthate
Hormone
Androgen
Synthetic depot
Testosterone propionate
Hormone
Androgen
Synthetic depot
Tetracaine
Local anaesthetic
Tetracycline
Antibiotic
Bacteriostatic protein synthesis inhibitor
Antiulcer
30S ribosome
Prevents aminoacyl tRNA attachment
Thalidomide
Antineoplastic
Anti-angiogenic
Anti-TNF
Theophylline
Bronchodilator
Methylxanthine
Phosphodiesterase inhibitor
Used in asthma
Thiabendazole
Antihelminthic
Treatment of intestinal roundworms
6-Thioguanine
Antineoplastic
Antimetabolite
(“pseudofeedback inhibition” of
HGPRT and PRP – purine synthesis)
Thiopental
General Anaesthetic
Ultra-short-acting barbiturate
Thioridazine
Antipsychotic
Phenothiazine
Thiotepa
Antineoplastic
Alkylating agent
Thiothixene
Antipsychotic
Thrombopoietin
Cytokine
Platelet synthesis stimulator
Thromboxane A2 (TXA2)
Autacoid
Promotes platelet aggregation
Cyclooxygenase product of
arachidonate metabolism
Thyrotropin-releasing
Hormone (TRH)
Hypothalamic hormone
Stimulates release of thyroid
stimulating hormone (TSH) from the
anterior pituitary
Thyrotropin
Thyroid-stimulating Hormone
(TSH)
Anterior pituitary hormone
Stimulates production of thyroxine
(T4), triiodothyronine (T3) and
thyroglobulin
Ticarcillin
Penicillin antibiotic
Cell wall synthesis inhibitor
Antiulcer
Anti-pseudomonal penicillin
Inhibits peptidoglycan cross-linking
Ticlopidine
Antiplatelet
ADP receptor antagonist
Timolol
Sympatholytic
 adrenergic antagonist
Antihypertensive
Glaucoma treatment
Anti-anginal
Bronchoconstrictor
Tissue plasminogen activators
alteplase, reteplase, tenecteplase
Thrombolytics
Tobramycin
Aminoglycoside antibiotic
Bactericidal protein synthesis inhibitor
30S ribosome
Freezes initiation
Tocainide
Class I antiarrhythmic
Na+ channel blocker
(activated channels)
Tolbutamide
Oral hypoglycemic
Sulfonylurea
Insulinotropic
Tolterodine
Anticholinergic
Muscarinic receptor antagonist
Prevents urination
Toremifene
Estrogen antagonist
Selective estrogen receptor
modulator (SERM)
Tosemide
Loop diuretic
Na-K-2Cl symporter inhibitor
Trandopril
Antihypertensive
Converting enzyme inhibitor
Tranylcypromine
Antidepressant
Monoamine oxidase inhibitor (MAO-I)
Trastuzumab
Antineoplastic
Anti-HER2 antibody
Triamcinolone
Adrenocorticosteroid
Glucocorticoid
Anti-inflammatory steroid
Inhaled
Triamterene
Potassium sparing diuretic
Sodium channel inhibitor
Antihypertensive
Triazolam
Sedative/Hypnotic
Benzodiazepine
Trifluoperazine
Antipsychotic
Phenothiazine
Trifluridine
Antiherpes
Pyrimidine analog
Phosphorylated to inhibitor of viral
DNA polymerase
Trihexyphenidyl
Antiparkinson
Antimuscarinic
Trimethaphan
Sympatholytic
Anticholinergic
Nicotinic antagonist
Antihypertensive
Trimethoprim
Antibiotic
Protein and nucleic acid
synthesis inhibitor
Folic acid antagonist
Inhibits bacterial dihydrofolate
reductase
Trimetrexate
Antibiotic
Folic acid antagonist
Treatment for Pneumocystis carinii
Tripelennamine
Classical antihistamine
H1 antagonist
Tubocurarine
Paralytic
Paralyzes skeletal muscles
Tumor necrosis factor 
Cytokine
Antineoplastic
Tyramine
Indirect sympathomimetic
Vasoconstrictor
Vasopressor
Ultralente insulin
Hormone
Insulin analogue
Long acting
Urokinase
Thrombolytic
Valacyclovir
Antiherpes
Purine analog
Phosphorylated to inhibitor of viral
DNA polymerase
Valdesartan
Antihypertensive
Angiotensin receptor blocker
(ARB)
Valganciclovir
Antiherpes
Purine analog
Phosphorylated to inhibitor of viral
DNA polymerase
Valproic acid
Anticonvulsant
Valsartan
Antihypertensive
Angiotensin receptor blocker
(ARB)
Vancomycin
Antibiotic
Inhibits cell wall synthesis
Not a  lactam
Arginine vasopressin
(Antidiuretic hormone; ADH)
Hypothalamic (posterior pituitary)
hormone
Antidiuretic
Vasoconstrictor
Vecuronium
Paralytic
Paralyze skeletal muscles
Verapamil
Class IV antiarrhythmic
Antihypertensive
L-type Ca2+ channel blocker
Antianginal
Vigabatrin
Anticonvulsant
Irreversible GABA aminotransferase
inhibitor
Vinblastine
Antineoplastic
Vinca alkaloid
Natural product
Vincristine
Antineoplastic
Vinca alkaloid
Natural product
Voriconazole
Triazole antifungal
Inhibits synthesis of ergosterol by
inhibiting lanosterol 14 demethylase
Warfarin
Anticoagulant
Vitamin K synthesis inhibitor
Zafirlukast
Leukotriene inhibitor
LTR1 and LTD4 antagonist
Asthma treatment
Zalcitabine
Antiretroviral
Nucleoside reverse transcriptase
inhibitor (NRTI)
Dideoxycytidine (ddC)
Zanamivir
Antiviral
Inhibits neuraminidase
and decreases viral release
Treatment of Influenza A & B
Zidovudine
Azidothymidine (AZT)
Antiretroviral
Nucleoside reverse transcriptase
inhibitor (NRTI)
Zileuton
Leukotriene inhibitor
5-lipoxygenase inhibitor
Used in asthma
Zolpidem
Sedative/Hypnotic
Non-benzodiazepine
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