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Table 1: Pharmacologic agents implicated in Drug-Induced Pseudolymphoma Syndrome and
Drug-Induced Hypersensitivity Syndrome.
Class
Antiarrhythmics
Antiarrhythmics
Antibiotics
Anticoagulants
Antidepressants
Antihistamines
Antihypertensives
Antipsychotics
Antirheumatics
Benzodiazepines
Chemotherapeutics
Reported Subclasses & Agents
Phenytoin, Carbamazepine, Butobarbital, Lamotrigine, Mephenytoin,
Methsuximide, Phenobarbital, Phensuximide, Primidone, Trimethadione,
Ethosuximide 2 *
Mexiletine, Procainamide
Flucloxacillin 2, Dapson, Cefixime, Nitrofurantoin, Penicillin, Sulfonamides
Fluinodione 2
Amitriptyline, Bupropion, Desipramine, Doxepin, Fluoxetine, Lithium,
Maprotiline
H1 blockers – Diphenhydramine
H2 blockers – Cimetidine, Ranitidine
Alpha agonists – Clonidine patch
Angiotensin-converting enzyme inhibitors – Benazepril, Captopril, Enalapril,
Lisinopril
Angiotensin receptor blockers – Losartan, Valsartan
Beta-blockers – Atenolol, Labetalol
Calcium channel blockers – Diltiazem, Verapamil
Diuretics – Hydrochlorothiazide, Hydrochlorothiazide with Amiloride
Vasodilators – Hydralazine
Phenothiazines – Chlorpromazine, Thioridazine, Promethazine
Allopurinol, D-penicillamine, Gold, Nonsteroidal Anti-Inflammatory Drugs
Clonazepam, Lorazepam
Cyclosporine, Methotrexate, Imatinib (Gleevac), Glatiramer acetate,
Oxaliplatin/5-fluorouracil/leucovorin1
Methylphenidate hydrochloride 12
Lovastatin
CNS stimulant
HMG-CoA reductase
inhibitors
Mast cell stabilizers
Cromolyn Sodium
Sex steroids
Estrogen, Progesterone
Topical agents
Etheric plant oil, Menthol, Hydroquinone cream 2
Vaccines
Hepatitis A or B vaccine injection sites
* References provided for agents added since last E-medicine publication
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