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Unofficial (P1) Year Drug List
Cardiac / Hypertension Drugs
ACEI (Angiotensin Converting Enzyme Inhibitor)
o
o
o
o
o
o
o
benazepril
captopril
enalapril
fosinopril
lisinopril
quinapril
ramipril
Lotensin®
Capoten®
Vasotec, Vaseretic®
Monopril®
Zestril®, Prinivil®
Accupril®
Altace®
Angiotensin II Receptor Antagonist
o irbesartan
o losartan
o valsartan
Beta-blocker
o
o
o
o
Avapro®
Cozaar®
Diovan®
(edited by s.fey)
Pharmacology
o Inhibit β1-receptors in SinoAtrial / AtrialVentricular node
o Decrease renin release
o Increase vasodilation
Efficacy
o Effective in lowering BP
o No proven reduction in Cardiovascular (CV) mortality
Side Effects
o Minor:
 confusion, lethargy, impotence, nightmares
 small increases in Triglyceride levels
 small decrease in HDL levels
o Major:
 Bradycardia, bronchiospasms, vasospasm
 Decreased tolerance to exercise
 Variations in blood glucose can mask hypoglycemia
 May aggravate CHF
Drugs, Doses, Half-Life, Brand Names (®)
o Atenolol
25 – 100 mg PO QD;
T1/2 = 3 – 4 hours
 Brand(s): Tenormin®
o Metoprolol
50 -100 mg PO QD;
T1/2 = 3 – 7 hours
 Brand(s): Toprol®, Lopressor®
o Propranolol
40 – 320 mg POQD;
T1/2 = 3 – 5 hours
 Brand(s): Inderal®
o Labetalol
100 – 200 PO BID;
T1/2 = 6 – 8 hours
 Brand(s): Normodyne®, Levatol®, Trandate®
o Carvedilol
6.25 – 25 mg PO QD, BID;
T1/2 = 7 – 10 hours
 Brand(s): Coreg
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Unofficial (P1) Year Drug List
Calcium Channel Blocker
o
o
o
o
amlodipine
diltiazem
nifedipine
verapamil
Norvasc®
Cardizem®
Procardia XL®, Adalat CC®
Calan, Calan SR®
Calcium Channel Blocker/ACEI
o amlodipine/benazepril
Lotrel®
Cardiac Glycoside
o digoxin
Lanoxin®
Diuretics
Loop Diuretics
o bumetanide
o furosemide
o torsemide
Bumex®
Lasix®
Demadex®
Potassium Sparing Diuretics
o spironolactone
Aldactone®
Potassium Sparing/Thiazide Diuretics
o triamterene/HCTZ Dyazide®
Thiazide Diuretics
o chlorthalidone
Hygroton®
o hydrochlorothiazide Hydrodiuril®
α1 Adrenergic Blocking Agent
o doxazosin
o terazosin
o clonidine
Cardura®
Hytrin®
Catapres®
Vasodilating Agents
o nitroglycerin (all forms)
Nitroquick®, Nitrolingual®
Miscellaneous
H2 Antagonists
o nizatidine
o famotidine
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Axid®
Pepcid®
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Unofficial (P1) Year Drug List
o cimetidine
o ranitidine
Tagamet®
Zantac®
Proton Pump inhibitors
o
o
o
o
Lansoprazole
Pantoprazole
Esomeprazole
Omeprazole
Prevacid®
Protonix®
Nexium®
Prilosec®
Antitussives, Expectorants, and Mucolytic Agents
o Dextromethorphan Benylin®
o Guaifenesin
Robitussin®
Sympathomimetic Agents
o Pseudoephedrine
Sudafed®
Analgesic/Antipyretic
o
o
o
o
aspirin
acetaminophen
ibuprofen
naproxen
Tylenol®, Excedrin®
Motrin®, Advil®, Nuprin®, Provel®
Pain Relievers
o hydrocodone
Lortab®, Lorcet®, Vicodin®
o fentanyl
Duragesic®
o acetaminophen with codeine
Tylenol® with codeine
Dyslipidemia
HMG CoA Reductase Inhibitors:
o
o
o
o
o
o
Atorvastatin
Simvastatin
Pravastatin
Rosuvastatin
Lovastatin
Fluvastatin
Lipitor®
Zocor®
Pravachol®
Crestor®
Mevacor®
Lescol®
Miscellaneous:
o Ezetimibe
Zetia®
Bile Acid Sequestrants:
o Cholestyramine
o Colestipol
o Colesevelam
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Questran®
Colestid®
WelChol™
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Unofficial (P1) Year Drug List
Nicotinic Acid Derivatives:
o Extended-release nicotinic acid
o Sustained-release nicotinic acid
o Crystalline nicotinic acid
Fibric Acid Derivatives:
o Gemfibrozil
o Fenofibrate
Lopid®
Tricor®
Combination Products:
o Ezetimibe / simvastatin
o Lovastatin / Niacin
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Vytorin®
Advicor®
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Niaspan®
Unofficial (P1) Year Drug List
Diabetes Drugs
Classification Brand Name Generic Names
o Sulfonylurea Diabeta/Micronase Glyburide
o Glucotrol
Glipizide
o Meglitinides Prandin
Repaglinide
o Starlix Nateglinide
o Biguanides Glucophage Metformin
o Thiazolidinediones Avandia Rosiglitazone
o Alpha-glucosidase Inhibitor
o Acarbose
Precose
o Insulins
Novolog
o Insulin
aspart
o Insulin
Humalog
lispro
o R Regular insulin Novolin R/Humulin
o N NPH insulin
isophane
Novolin N/Humulin
o Insulin
glargine Lantus
Mechanisms of Action
o Sulfonlyureas – stimulate insulin release from pancreatic beta-cells
o Meglitinides – stimulate insulin release from pancreatic beta-cells
o Biguanides – decreases glucose output from the liver & increases peripheral
muscle glucose uptake
o Thiazolidinediones (TZD) – decrease peripheral (skeletal muscle and adipose
tissue) insulin resistance & decreases hepatic glucose production
o Alpha-glucosidase Inhibitors – decreases the breakdown of carbohydrates in
the brush border of the small intestine
o Insulin – recombinant DNA insulin that replaces endogenously produced insulin
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Unofficial (P1) Year Drug List
Antibiotics Community related drugs
o
o
o
o
o
o
o
o
o
o
o
o
o
o
o
o
o
o
o
o
Diflucan®
Valtrex®
Omnicef®
Amoxil®
Augmentin
Zithromax®
Biaxin®
Cefzil®
Levaquin®
Tequin®
Avelox®
Cipro®
Tamiflu®
Macrobid
Doxycycline
Tetracycline
Minocin®
Flagyl®
Penicillin
Bactrim®
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Unofficial (P1) Year Drug List
Asthma Drug List
Prescription Rescue β-agonists
o Albuterol (Proventil HFA/Ventolin)
o Pirbuterol (Maxair Autohaler)
Anticholinergics
o Ipratropium:
o Ipratropium & Albuterol
o Ipratropium
Combivent
Atrovent
Systemic Corticosteroids
o Methylprednisolone (DosePak only)
o Prednisone Tablets
Long Term Controllers
o β-agonists
o Salmeterol
Serevent Inhaler
Inhaled Corticosteroids
o
o
o
o
o
o
o
o
o
o
Budesonide
Rhinocort
Beclomethasone
Beclomethasone MDI and nasal Vancenase, Vancenase AQ/Beconase,
Vanceril/Beclovent)
Beclomethasone diproprionate HFA
Qvar
Fluticasone & Salmeterol Advair
Fluticasone
Flonase
Fluticasone
Flovent
Mometasone Furoate Monohydrate
Nasonex
Triamcinolone
Azmacort
Leukotriene Modifiers
o Montelukast
o Zafirlukast
Singulair
Accolate
Mast Cell Stabilizers
o Cromolyn
Intal
Inhaled Anticholinergics
o Tiotropium
Spiriva
Miscellaneous
o Theophylline (various types and names)
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Unofficial (P1) Year Drug List
Antihistamines
o Cetirizine
o Fexofenadine
o Loratadine
Zyrtec®
Allegra®
Claritin®, various
OTC
o Clemastine
o Loratadine
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Tavist®
Claritin®
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Unofficial (P1) Year Drug List
Controlled Substance Drug Schedules
SCHEDULE I – Drugs that have no currently accepted medical use in treatment in
The United States and have a high potential for abuse. The average
practitioner may not prescribe Schedule I drugs.
Examples:
o Opiates, Opium derivatives such as Heroin
o Hallucinogens (LSD)
o Marijuana
o Depressants such as: Methaqualone (Quaalude®)
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Unofficial (P1) Year Drug List
SCHEDULE II – Drugs that have a high potential for abuse and have a currently
accepted medical use in treatment in the United States or a currently
accepted medical use with severe restrictions.
Generic or Chemical Name Brand or Proprietary Name
o Alfentanil
Alfenta
o Amobarbital
Amytal, Tuinal
o Amphetamine
Dexedrine, Adderall
o Belladonna w/Opium B&O Suppositories
o Cocaine
Various manufacturers
o Fentanyl
Duragesic, Actiq
o Hydromorphone
Dilaudid
o Meperidine
Demerol
o Methadone
Dolophine, Methadose, Amidone
o Methylphenidate
Ritalin, Concerta, Metadate, Metadate CD
o Morphine
MS Contin, MSIR, Roxanol, Duramorph
o Oxycodone
OxyContin®, Roxicodone,
o With APAP
Percocet, Roxicet,
o Tylox,
Endocet
o With ASA Percodan,
Endodan
o Oxymorphone
Numorphan
o Pentobarbital
Nembutal
o Remifentanil
Ultiva
o Secobarbital
Seconal, Tuinal
o Sufentanil
Sufenta
SCHEDULE II NYS
SCHEDULE III FEDERAL ANABOLIC STEROIDS
Generic or Chemical Name Brand or Proprietary Name
o Dihydrotestosterone
Stanolone
o Ethylestrenol
Maxibolin, Orabolin
o Fluoxymesterone
Android-F, Halotestin
o Methandrostenolone
Dianabol
o Methyltestosterone
Anadroid
o Nandrolone
Decanoate Deca-Durabolin
o Nandrolone
Phenpropionate Durabolin
o Oxandrolone
Anavar, Lonavar, Provitar
o Oxymetholone
Anadrol-50
o Stanolone
Anabolex
o Stanozolol
Winstrol
o Testosterone
Android-T, Androlan, Depotest, Delatestryl
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Unofficial (P1) Year Drug List
SCHEDULE III – Drugs that have a potential for abuse less than the drugs in
Schedule I and II and have a currently accepted medical use in the
United States.
Generic or Chemical Name Brand or Proprietary Name
o Acetaminophen with Codeine
Tylenol® with Codeine
o Amobarbital suppository
Amytal
o Aspirin with Butalbital and Codeine Fiorinal with Codeine
o Aspirin with Codeine
Empirin with Codeine
o Aspirin with Butalbital
Fiorinal
o Buprenorphine F = III S =V Subutex, Suboxone, Buprenex, Temegesic
o Dronabinol
Marinol
o Hydrocodone Combinations:
o With Chlorpheniramine
Tussionex
o With APAP
Lortab, Vicodin
o With ASA
Lortab ASA
o With Guaifenesin
Hycotuss, Vicodin Tuss
o With Ibuprofen
Vicoprofen
o Ketamine
Ketalar
o Paregoric Liquid
Various manufacturers
o Pentobarbital Suppository Nembutal
o Phendimetrazine
Plegine, Bontril, Prelu-2
o Secobarbital Suppository Seconal
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Unofficial (P1) Year Drug List
SCHEDULE IV – Drugs that have a low potential for abuse relative to the drugs in
Schedule III with a currently accepted medical use in the United States.
Generic or Chemical Name
Brand or Proprietary Name (®)
o Butorphanol (Federal Control IV only) Stadol
o Chloral Hydrate
Noctec®, Aquachloral®
o Dichloralphenazone
Midrin
o Meprobamate
Miltown, Equanil, Deprol
o Modafinil
Provigil
o Pemoline
Cylert
o Pentazocine
Talwin NX, Talacen, Talwin Compound
o Phenobarbital
Various manufacturers
o Phentermine
Adipex-P, Ionamin
o Propoxyphene
Darvon
o With APAP
Darvocet, Darvocet N-100
o With ASA
Darvon Compound
o Sibutramine
Meridia
o Zaleplon
Sonata
o Zolpidem
Ambien
SCEHDULE IV BENZODIAZEPINES
Generic or Chemical Name Brand or Proprietary Name
o Alprazolam
Xanax
o Chlordiazepoxide
Librium, Libritabs
o Chlordiazepoxide & methoscopolamine
Librax
o Clonazepam
Klonopin
o Clorazepate
Tranxene
o Diazepam
Valium
o Estazolam
ProSom
o Fluitrazepam
Rohypnol (Not available in US)
o Flurazepam
Dalmane
o Lorazepam
Ativan
o Midazolam
Versed
o Oxazepam
Serax
o Temazepam
Restoril
o Triazolam
Halcion
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Unofficial (P1) Year Drug List
SCHEDULE V – Drugs that have a low potential for abuse relative to the drugs in
Schedule IV with a currently accepted medical use in the United States.
Generic or Chemical Name Brand or Proprietary Name
o Codeine cough syrups Robitussin AC (Guaifenesin)
o Guiatuss AC, Mytussin AC, Cheracol
o Diphenoxylate/Atropine Lomotil
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