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Unofficial (P1) Year Drug List Cardiac / Hypertension Drugs ACEI (Angiotensin Converting Enzyme Inhibitor) o o o o o o o benazepril captopril enalapril fosinopril lisinopril quinapril ramipril Lotensin® Capoten® Vasotec, Vaseretic® Monopril® Zestril®, Prinivil® Accupril® Altace® Angiotensin II Receptor Antagonist o irbesartan o losartan o valsartan Beta-blocker o o o o Avapro® Cozaar® Diovan® (edited by s.fey) Pharmacology o Inhibit β1-receptors in SinoAtrial / AtrialVentricular node o Decrease renin release o Increase vasodilation Efficacy o Effective in lowering BP o No proven reduction in Cardiovascular (CV) mortality Side Effects o Minor: confusion, lethargy, impotence, nightmares small increases in Triglyceride levels small decrease in HDL levels o Major: Bradycardia, bronchiospasms, vasospasm Decreased tolerance to exercise Variations in blood glucose can mask hypoglycemia May aggravate CHF Drugs, Doses, Half-Life, Brand Names (®) o Atenolol 25 – 100 mg PO QD; T1/2 = 3 – 4 hours Brand(s): Tenormin® o Metoprolol 50 -100 mg PO QD; T1/2 = 3 – 7 hours Brand(s): Toprol®, Lopressor® o Propranolol 40 – 320 mg POQD; T1/2 = 3 – 5 hours Brand(s): Inderal® o Labetalol 100 – 200 PO BID; T1/2 = 6 – 8 hours Brand(s): Normodyne®, Levatol®, Trandate® o Carvedilol 6.25 – 25 mg PO QD, BID; T1/2 = 7 – 10 hours Brand(s): Coreg 582750849 Page 1 Unofficial (P1) Year Drug List Calcium Channel Blocker o o o o amlodipine diltiazem nifedipine verapamil Norvasc® Cardizem® Procardia XL®, Adalat CC® Calan, Calan SR® Calcium Channel Blocker/ACEI o amlodipine/benazepril Lotrel® Cardiac Glycoside o digoxin Lanoxin® Diuretics Loop Diuretics o bumetanide o furosemide o torsemide Bumex® Lasix® Demadex® Potassium Sparing Diuretics o spironolactone Aldactone® Potassium Sparing/Thiazide Diuretics o triamterene/HCTZ Dyazide® Thiazide Diuretics o chlorthalidone Hygroton® o hydrochlorothiazide Hydrodiuril® α1 Adrenergic Blocking Agent o doxazosin o terazosin o clonidine Cardura® Hytrin® Catapres® Vasodilating Agents o nitroglycerin (all forms) Nitroquick®, Nitrolingual® Miscellaneous H2 Antagonists o nizatidine o famotidine 582750849 Axid® Pepcid® Page 2 Unofficial (P1) Year Drug List o cimetidine o ranitidine Tagamet® Zantac® Proton Pump inhibitors o o o o Lansoprazole Pantoprazole Esomeprazole Omeprazole Prevacid® Protonix® Nexium® Prilosec® Antitussives, Expectorants, and Mucolytic Agents o Dextromethorphan Benylin® o Guaifenesin Robitussin® Sympathomimetic Agents o Pseudoephedrine Sudafed® Analgesic/Antipyretic o o o o aspirin acetaminophen ibuprofen naproxen Tylenol®, Excedrin® Motrin®, Advil®, Nuprin®, Provel® Pain Relievers o hydrocodone Lortab®, Lorcet®, Vicodin® o fentanyl Duragesic® o acetaminophen with codeine Tylenol® with codeine Dyslipidemia HMG CoA Reductase Inhibitors: o o o o o o Atorvastatin Simvastatin Pravastatin Rosuvastatin Lovastatin Fluvastatin Lipitor® Zocor® Pravachol® Crestor® Mevacor® Lescol® Miscellaneous: o Ezetimibe Zetia® Bile Acid Sequestrants: o Cholestyramine o Colestipol o Colesevelam 582750849 Questran® Colestid® WelChol™ Page 3 Unofficial (P1) Year Drug List Nicotinic Acid Derivatives: o Extended-release nicotinic acid o Sustained-release nicotinic acid o Crystalline nicotinic acid Fibric Acid Derivatives: o Gemfibrozil o Fenofibrate Lopid® Tricor® Combination Products: o Ezetimibe / simvastatin o Lovastatin / Niacin 582750849 Vytorin® Advicor® Page 4 Niaspan® Unofficial (P1) Year Drug List Diabetes Drugs Classification Brand Name Generic Names o Sulfonylurea Diabeta/Micronase Glyburide o Glucotrol Glipizide o Meglitinides Prandin Repaglinide o Starlix Nateglinide o Biguanides Glucophage Metformin o Thiazolidinediones Avandia Rosiglitazone o Alpha-glucosidase Inhibitor o Acarbose Precose o Insulins Novolog o Insulin aspart o Insulin Humalog lispro o R Regular insulin Novolin R/Humulin o N NPH insulin isophane Novolin N/Humulin o Insulin glargine Lantus Mechanisms of Action o Sulfonlyureas – stimulate insulin release from pancreatic beta-cells o Meglitinides – stimulate insulin release from pancreatic beta-cells o Biguanides – decreases glucose output from the liver & increases peripheral muscle glucose uptake o Thiazolidinediones (TZD) – decrease peripheral (skeletal muscle and adipose tissue) insulin resistance & decreases hepatic glucose production o Alpha-glucosidase Inhibitors – decreases the breakdown of carbohydrates in the brush border of the small intestine o Insulin – recombinant DNA insulin that replaces endogenously produced insulin 582750849 Page 5 Unofficial (P1) Year Drug List Antibiotics Community related drugs o o o o o o o o o o o o o o o o o o o o Diflucan® Valtrex® Omnicef® Amoxil® Augmentin Zithromax® Biaxin® Cefzil® Levaquin® Tequin® Avelox® Cipro® Tamiflu® Macrobid Doxycycline Tetracycline Minocin® Flagyl® Penicillin Bactrim® 582750849 Page 6 Unofficial (P1) Year Drug List Asthma Drug List Prescription Rescue β-agonists o Albuterol (Proventil HFA/Ventolin) o Pirbuterol (Maxair Autohaler) Anticholinergics o Ipratropium: o Ipratropium & Albuterol o Ipratropium Combivent Atrovent Systemic Corticosteroids o Methylprednisolone (DosePak only) o Prednisone Tablets Long Term Controllers o β-agonists o Salmeterol Serevent Inhaler Inhaled Corticosteroids o o o o o o o o o o Budesonide Rhinocort Beclomethasone Beclomethasone MDI and nasal Vancenase, Vancenase AQ/Beconase, Vanceril/Beclovent) Beclomethasone diproprionate HFA Qvar Fluticasone & Salmeterol Advair Fluticasone Flonase Fluticasone Flovent Mometasone Furoate Monohydrate Nasonex Triamcinolone Azmacort Leukotriene Modifiers o Montelukast o Zafirlukast Singulair Accolate Mast Cell Stabilizers o Cromolyn Intal Inhaled Anticholinergics o Tiotropium Spiriva Miscellaneous o Theophylline (various types and names) 582750849 Page 7 Unofficial (P1) Year Drug List Antihistamines o Cetirizine o Fexofenadine o Loratadine Zyrtec® Allegra® Claritin®, various OTC o Clemastine o Loratadine 582750849 Tavist® Claritin® Page 8 Unofficial (P1) Year Drug List Controlled Substance Drug Schedules SCHEDULE I – Drugs that have no currently accepted medical use in treatment in The United States and have a high potential for abuse. The average practitioner may not prescribe Schedule I drugs. Examples: o Opiates, Opium derivatives such as Heroin o Hallucinogens (LSD) o Marijuana o Depressants such as: Methaqualone (Quaalude®) 582750849 Page 9 Unofficial (P1) Year Drug List SCHEDULE II – Drugs that have a high potential for abuse and have a currently accepted medical use in treatment in the United States or a currently accepted medical use with severe restrictions. Generic or Chemical Name Brand or Proprietary Name o Alfentanil Alfenta o Amobarbital Amytal, Tuinal o Amphetamine Dexedrine, Adderall o Belladonna w/Opium B&O Suppositories o Cocaine Various manufacturers o Fentanyl Duragesic, Actiq o Hydromorphone Dilaudid o Meperidine Demerol o Methadone Dolophine, Methadose, Amidone o Methylphenidate Ritalin, Concerta, Metadate, Metadate CD o Morphine MS Contin, MSIR, Roxanol, Duramorph o Oxycodone OxyContin®, Roxicodone, o With APAP Percocet, Roxicet, o Tylox, Endocet o With ASA Percodan, Endodan o Oxymorphone Numorphan o Pentobarbital Nembutal o Remifentanil Ultiva o Secobarbital Seconal, Tuinal o Sufentanil Sufenta SCHEDULE II NYS SCHEDULE III FEDERAL ANABOLIC STEROIDS Generic or Chemical Name Brand or Proprietary Name o Dihydrotestosterone Stanolone o Ethylestrenol Maxibolin, Orabolin o Fluoxymesterone Android-F, Halotestin o Methandrostenolone Dianabol o Methyltestosterone Anadroid o Nandrolone Decanoate Deca-Durabolin o Nandrolone Phenpropionate Durabolin o Oxandrolone Anavar, Lonavar, Provitar o Oxymetholone Anadrol-50 o Stanolone Anabolex o Stanozolol Winstrol o Testosterone Android-T, Androlan, Depotest, Delatestryl 582750849 Page 10 Unofficial (P1) Year Drug List SCHEDULE III – Drugs that have a potential for abuse less than the drugs in Schedule I and II and have a currently accepted medical use in the United States. Generic or Chemical Name Brand or Proprietary Name o Acetaminophen with Codeine Tylenol® with Codeine o Amobarbital suppository Amytal o Aspirin with Butalbital and Codeine Fiorinal with Codeine o Aspirin with Codeine Empirin with Codeine o Aspirin with Butalbital Fiorinal o Buprenorphine F = III S =V Subutex, Suboxone, Buprenex, Temegesic o Dronabinol Marinol o Hydrocodone Combinations: o With Chlorpheniramine Tussionex o With APAP Lortab, Vicodin o With ASA Lortab ASA o With Guaifenesin Hycotuss, Vicodin Tuss o With Ibuprofen Vicoprofen o Ketamine Ketalar o Paregoric Liquid Various manufacturers o Pentobarbital Suppository Nembutal o Phendimetrazine Plegine, Bontril, Prelu-2 o Secobarbital Suppository Seconal 582750849 Page 11 Unofficial (P1) Year Drug List SCHEDULE IV – Drugs that have a low potential for abuse relative to the drugs in Schedule III with a currently accepted medical use in the United States. Generic or Chemical Name Brand or Proprietary Name (®) o Butorphanol (Federal Control IV only) Stadol o Chloral Hydrate Noctec®, Aquachloral® o Dichloralphenazone Midrin o Meprobamate Miltown, Equanil, Deprol o Modafinil Provigil o Pemoline Cylert o Pentazocine Talwin NX, Talacen, Talwin Compound o Phenobarbital Various manufacturers o Phentermine Adipex-P, Ionamin o Propoxyphene Darvon o With APAP Darvocet, Darvocet N-100 o With ASA Darvon Compound o Sibutramine Meridia o Zaleplon Sonata o Zolpidem Ambien SCEHDULE IV BENZODIAZEPINES Generic or Chemical Name Brand or Proprietary Name o Alprazolam Xanax o Chlordiazepoxide Librium, Libritabs o Chlordiazepoxide & methoscopolamine Librax o Clonazepam Klonopin o Clorazepate Tranxene o Diazepam Valium o Estazolam ProSom o Fluitrazepam Rohypnol (Not available in US) o Flurazepam Dalmane o Lorazepam Ativan o Midazolam Versed o Oxazepam Serax o Temazepam Restoril o Triazolam Halcion 582750849 Page 12 Unofficial (P1) Year Drug List SCHEDULE V – Drugs that have a low potential for abuse relative to the drugs in Schedule IV with a currently accepted medical use in the United States. Generic or Chemical Name Brand or Proprietary Name o Codeine cough syrups Robitussin AC (Guaifenesin) o Guiatuss AC, Mytussin AC, Cheracol o Diphenoxylate/Atropine Lomotil 582750849 Page 13