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Poster Session B
P116
G.P. Bandopadhyaya, J. Shukla, R. Kumar, A.Malhotra
Designing radiolabelled DMSA loaded PLGA microspheres: an experimental
module for targeted radiotherapy using Glioma cell line
P117
M. Niemyjska,D. Maciejewska, M. Włostowski, M. Żemajtys
Syntheses and structural analyses of 3,3-diindolilomethane derivatives, potential
inhibitors of cell proliferation in human breast cancer cells
P118
K. Studzian, M. Wąsowska, E. Ciesielska, I. Oszczapowicz, L. Szmigiero
Studies on the mechanism of cytotoxic action of new daunorubicin analogue
P119
M. Wąsowska, J. Oszczapowicz, I. Oszczapowicz, J. Wietrzyk, A. Opolski,
A. Nasulewicz
Overcoming drug resistance of cancer cells by new group of anthracycline
antibiotics
P120
A. Bielawska, K. Bielawski, A. Muszyńska, T. Anchim
Role of DNA binding and inhibition of human DNA topoisomerase II in cytotoxicity
of novel amidine analogues of chlorambucil in breast cancer MCF-7
P121
K. Bielawski, A. Bielawska, K. Kosk, S. Wołczyński
Synthesis, DNA binding, and biological evaluation of bisbenzimidazole derivatives
with alkylating moiety
P122
J. Kossakowski, E. Hejchman, K. Ostrowska
Synthesis of new derivatives of benzofuran-2 and benzofuran-3-carboxylic acid with
potential anticancer activity
P123
P. Diana, A. Martorana, P. Barraja, A. Lauria, A. Montalbano, A.M. Almerico,
G. Dattolo, G. Cirrincione
Isoindolo[1,2-a]quinoxalin-4(5H)-one: a new ring system with potential antitumor
activity
P124
Joanna Cytarska, Marek Zaidlewicz
Synthesis of a cyclobutane analogue of BPA for boron neutron capture therapy
P125
A. Wiosetek-Reske, S. Wysocki
Investigation of spectral properies of the intercalation complex between n-nonylacridine orange and DNA
P126
J. Wietrzyk, B. Filip, A. Trzeciakiewicz, A. Kutner, W. Szelejewski, A. Opolski
Calcitriol down-regulates β3 integrins expression and suppresses the malignant
phenotype in a Lewis lung carcinoma cell line
P127
I. Jaroszewicz, M. Pełczyńska, A. Kutner, W. Szelejewski, A. Opolski
The correlation between nVDR expression and antiproliferative activity of calcitriol
or its new analogues against various tumor cell lines
P128
J. Sławiński
Synthesis of a new series of 4-chloro-2-mercapto-5-methylbenzene-sulfonamide
derivatives with potential antitumor activity
P129
C. Bolchi, R. Di Pumpo, L. Fumagalli, M. Pallavicini, A. Pedretti, E. Valoti,
L. Villa, G. Vistoli
Design, synthesis and biological evaluation of non-peptidic inhibitors of
farnesyltransferase
P130
K. Gąsiorowski, W. Malinka, P. Świątek, A. Jaszczyszyn
Antimutagenic activity of new analogues of fluphenazine
P131
G. Dormán, F. Darvas, L. Ürge, Á. Papp, M. Sasvári-Székely, I. Sziráki
Design and discovery of novel dopamine transporter inhibitors
P132
D. Posselt, R. Gust
Cytotoxicity and anti-tumour activity of novel iron Schiff´s base complexes
P133
S. Sobiak, M. Wierzchowski
Synthesis and conformational analysis of 3-(5-bromo-2-methyl-4-nitro-1H-imidazol1-yl)-1-(4-halogenophenyl)propane-1,2-dione
P134
S. Sobiak, M. Wieczorek, M. Wierzchowski
Synthesis of anticancer preventive mercaptoderivatives of trans-stilbene
P135
S. Małycha, L. Zaprutko
A comparison of conformational changes in some phthalideisoquinoline derivatives
P136
U. Kalinowska
Preparation, characterization and cytotoxicity evaluation of the novel platinum (II)
and palladium (II) complexes with phosphoric acid diethyl ester pyridinylmethyl
ester isomers. X-ray crystal structure of trans-dichlorobis(diethyl pyridin-2ylmethylphoshpate-кN)palladium(II)
P137
K. Aranowska, L. Szmigiero, J. Ochocki
Cis-(bispyridinylmethylphosphonate)platinum(II) complexes – spectroscopy,
structure and in vitro cytostatic activity
P138
M. Incerti, C.A. Maggiali, G. Morini, P. Vicini, R. Loddo, M. Saddi, R. Garijo,
M. Mura
Evaluation of the antiproliferative activity of benzofused nitrogen and sulfur/oxygen
containing heterocycles derivatives
P139
R. Ottanà, R. Maccari, G. Chiricosta, S. Cuzzocrea, S. Carotti, M. L. Barreca,
M.G. Vigorita
Design and synthesis of 5-aryliden-2-imino-4-thiazolidinones celecoxib analogues
as antiinflammatory and anticancer agents
P140
A.M. Panico, V. Cardile, R. Morrone, G. Nicolosi, B. Gentile, G. Ronsisvalle
(R) and (S) ketoprofen inhibit DU 145 and HELA cells growth
P141
A.M. Panico, M. Incerti, M. Mor, P. Vicini, F. Garufi, G Ronsisvalle
Synthesis and anticancer activity of new amidinobenzisothiazoles
P142
J. Achremowicz, A. Galanty, Z. Janeczko
Betulin derivatives as potent chemotherapeutics
P143
M. Sieńczyk, J. Oleksyszyn
New inhibitors for urokinase type plasminogen activator
P144
C. Campestre, S. Preziuso, M. Agamennone, P. Tortorella, C. Gallina
Synthesis and biological evaluation of new matrix metalloproteinases inhibitors
P145
A. Jezierska, M. Mączyński, S. Ryng
5-Substituted 3-methylisoxazole[5,4-d]1,2,3-triazin-4-one derivatives: synthesis and
computational study of immunologically active compounds
P146
P. La Colla, M.A. Piano, B. Poddesu, F. Marturana, G. Rassu, L. Auzzas,
V. Zambrano, L. Pinna, C. Curti
Synthesis and biological activity of carbasugar derivatives
P147
T. Ostrowski, B. Golankiewicz, E. De Clercq, J. Balzarini
Fluoro-substitution and 7-alkylation / arylalkylation as prospective modifications of
biologically active 6-aryl derivatives of TACV and TGCV
P148
A. Carta, C. Congiatu, M. Loriga, E. Marongiu, F. Esposito, R. Loddo
Synthesis and biological evaluation of N-[4-(1(2)H(benzotriazol-1(2)yl)phenylalkylcarboxamido and N,N’-bis-[4-1(2)H(benzotriazol-1(2)yl)phenylalkyldicarboxamido derivatives
P149
I. Weidlich, A. Matschay, S. Sobiak
Synthesis and study of SAR for 2-(1-adamantyl)imidazo[1,2-a]pyridine
and 2-(1-adamantyl)imidazo[1,2-a]pyrimidine derivatives using semiempirical
calculation by Hyperchem Professional
P150
M. Sechi, L. Sannia, M. Derudas, F. Carta, M. Orecchioni, R. Dallocchio,
A. Dessì, T. Sanchez, N. Neamati
Design, synthesis, structural investigation, docking studies and biological activities
of substituted-isoxazole carboxylic acids as HIV-1 integrase inhibitors
P151
M. Sechi, F. Carta, L. Sannia, M. Derudas, M. Palomba, R. Dallocchio,
A. Dessì, T. Sanchez, N. Neamati
Search for selective HIV-1 integrase inhibitors
P152
L. Mina, B. Tasso, C. Canu Boido, V. Boido, F. Sparatore, M. Marongiu,
C. A. Cabras, G. Collu, G. Pinna Spada, P. La Colla
Antiviral activity of variously substituted benzoazoles
P153
O. Tabarrini, G. Manfroni, A. Fravolini, V. Cecchetti, S. Sabatini, J. Paeshuyse,
E. De Clercq, J. Neyts
Selective anti-BVDV acridones as new potential anti-HCV agents
P154
R. Lisiak, M. Osajda, M. Chojnacka J. Palus, E. Piasecki, K. Rybka
Benzisoselenazolones and diselenides with polyamine moieties a new class of
antiviral agents
P155
J. Matysiak, A. Niewiadomy, R. Czeczko
Synthesis and in vitro antimycotic activity of 2-(2,4-dihydroxyphenyl)benzoxazoles
P156
S. Aiello, E. Aiello, M. Milici
Synthesis and antifungal activity of new 3(5)-methyl-5(3)-(2-thiophenyl)
and –(2-quinolyl)-1H-1-R-4-nitrosopyrazoles. Part V
P157
R. Fringuelli, F. Schiaffella, A. Macchiarulo, L. Milanese, G. Costantino,
D. Pietrella, A. Vecchiarelli
1,4-Benzothiazine and 1,4-benzoxazine imidazole derivatives with antifungal
activity
P158
B. Modzelewska-Banachiewicz, J. Kutkowska, Z. Zwolska, T. Urbanik,
W. Rzeski
Synthesis and biological activity of 3,4-disubstituted-1,2,4-triazole derivatives
P159
J. Cieplik, J. Pluta, O. Gubrynowicz
Synthesis and antimicrobial properties 3-sulfonyl-1,2,3,4-tetrahydropyrimido[4,5-d]pyrimidine derivatives
P160
A. Matschay, S. Sobiak, I. Weidlich
Synthesis 6-chloro-5-sulfamoylo-4-quinazolinone derivatives /Part 2/
P161
R. Maccari, R. Ottanà, E. Rotondo, C. Curinga, M.G. Vigorita
In vitro antimycobacterial activity of isoniazid-related metalchelates
P162
K. Amssoms, A. Yamani, A.-M. Lambeir, S.L. Oza, A.H. Fairlamb,
K. Augustyns, A. Haemers
Trypanothione synthesis as target in the design of antitrypanosomal agents
P163
Ł. Glinka, E. Nawrot, E. Zyner, E. Szewczyk, J. Ochocki
Synthesis and bacteriological activity of substituted flavonoid system – containing
ligands
P164
M. Pitucha, M. Dobosz, U. Kosikowska
Synthesis and biological action of 1-[(4-phenylpiperazinyl)methyl]-3-R-4-phenylΔ2-1,2,4-triazoline-5-thione
P165
M. Giurg, I. Maliszewska, K. Markiewicz, P. Podolski
Antimicrobial activity of halogen derivatives of 5-alkyl-3-aryl-1,2,4-oxadiazoles
P166
B. Vanderhoydonck, C.V. Stevens
Synthesis of phosphono gamma lactams from 1-phosphono-2-aza-1,3-dienes
P167
M. Hussein, T. Aboul-Fadl, A. Abdel-Nasser
Synthesis and antitubercular activity of some Schiff bases derived from Mannich
bases of isatin and isonicotinic acid hydrazide (INH)
P168
M. Agamennone, A. Tafi, C. Gallina, M. Botta
Amber* force field implementation to dock alkyl and aryl boronic acids as
β-lactamases inhibitors
P169
S. Preziuso, C. Campestre, M. Agamennone, P. Tortorella, G. Amicosante,
C. Gallina
Derivatives of m-aminophenylboronic acid as β-lactamases inhibitors
P170
K. Kieć-Kononowicz, E. Szymańska
Is (un)substituted sulphur necessary for antimycobacterial activity of arylidene
(thio)hydantoins?
P171
E. Szymańska, K. Kieć-Kononowicz
Analysis of physicochemical and topological properties among 5-arylidene
derivatives of hydantoin with antitubercular activity
P172
J. Janiszewska, A.W. Lipkowski, Z. Urbańczyk-Lipkowska
Rational design of antimicrobial peptide dendrimers
P173
G. Cardillo, L. Gentilucci, A. Tolomelli, M. Calienni, A. Qasem, S. Spampanato
Opioid peptide analogues containing β-Pro show antinociceptive activity after
periphereal administration
P174
F. Tóth, J. Farkas, G. Tóth, A. Borsodi, S. Benyhe
Synthesis, binding characteristics and G-protein activation of a novel synthetic
Met-enkephalin-Arg-Phe analogue
P175
J. Farkas, R. Guerrini, S. Salvadori, G. Orosz, G. Tóth
Preparation of the new tritiated nociceptin analogues. Study of the degradation
process
R. Löser, K. Schilling, M. Gütschow
Interaction of papain and papain-like cysteine proteases with dipeptide-derived
nitriles
P176
P177
R. Ostaszewski, A. Fryszkowska
Application of one - pot enzymatic desymmetrization and ugi MCR to the synthesis
of chiral peptidomimetics
P178
B. Leitgeb, A. Szekeres, G. Tóth
Conformational analysis of endomorphins by simulated annealing
P179
A.W. Lipkowski, P. Kosson, A. Misicka, Z. Lipkowska, G. Ronsisvalle,
D.B. Carr
Mimetic of opioid tyramine active conformation
P180
S. Weyler, A. Hunder, M. Kaulich, C.E. Müller
Combinatorial synthesis of acid blue 25 derivatives as P2Y 2 receptor antagonists
P181
A. Arany, A. Stevens, B. Vickery, C. Lauret, D. Boumrah, L. Phillips,
N. Church, J. Mankee, J. Harris, O. Olivera, R. Lau, S. Yau, S. Edwards
Tyrosine and serine / threonine targeted SoftFocus TM Libraries; design and
synthesis
P182
I. Weidlich, S. Sobiak
Merifield solid support nitroimidazole derivatives of nitrogen mustard synthesis
P183
R. Ostaszewski, W. Kurek
A new method of the synthesis of arginine peptidomimetics
P184
J. Turło, O. Lubiński, B. Gutkowska, A. Błażewicz, R. Kocjan
Submerged cultivation of Lentinus edodes on selenium enriched media
P185
A. Bartmańska, J. Dmochowska-Gładysz, A. Szpineter
Testolactones – products of biotransformation
P186
A. Szpineter, T. Kołek, A. Świzdor
7α-Hydroxy-dehydroepiandrosterone levels in culture of fungi Absidia coerulea
treated with phenobarbital
P187
A. Godawska, E. Pękala, K. Kieć-Kononowicz
Biotransformation of Praziquantel in silico
P188
S.S. Kamaeva, L.A. Potselueva, N.L. Zshavoroncova
The study of Aethonium release from the ointment by the microbiological method
P189
G.U. Mercureva, L.A. Potselueva, N.M. Aschurbaeva, S.B. Bogdanova
The study of ointment base influence on the honey antimicrobial activity
P190
M. Přádný, P. Lesný, J. Michálek, E. Sykováand, J. Vacík
Macroporous hydrogels based on copolymers of 2-hydroxyethyl methacrylate with
positively and/or negatively charged comonomers for implants into the CNS
P191
Yu.A. Egoshina, R.Sh. Valiev, L.A. Potselueva, T.N. Galiullina
Installation of an optimum of quantitative ratio the combination of isoniazid and
rifampicin in experience "in vitro"
P192
W. Marcoin
Influence of the selected auxiliary substances on the absorption process of Mg 2+ ions
from solid dispersions containing magnesium salts
P193
K. Majewska, L. Zaprutko
Microwave assisted synthesis of laurocapram (Azone)
P194
L. Zaprutko, D. Partyka B. Bednarczyk–Cwynar
New triterpenoid thiolactams as transdermal penetration enhancers
P195
P. Jaiswal, I.C. Shukla
Application of N-bromosuccinimide for determination of alkylating agents in pure
and pharmaceutical preparations
P196
J. Michalik, U. Karczmarczyk, A. Markiewicz
Comparative evaluation of 99m Tc-HYNIC-hIgG with EDTA as chelating agent.
Serum stability improvement in presence of divalent cations
P197
S. Kolp, M. Pietsch, E. A. Galinski, M. Gütschow
Protection against proteolytic cleavage by compatible solutes
P198
I. Muszalska, H. Śladowska, D. Szkatuła
HPLC and TLC methodology for determination and purity of 4-methoxy2-[2-hydroxy-3(4-phenyl-1-piperazinyl)]propyl-2,3-dihydro-6-methyl-1,3-dioxo1H-pyrrolo[3,4-c]pyridine
P199
I. Muszalska, H. Śladowska, D. Szkatuła
Kinetic studies of the degradation of 4-methoxy-2-[2-hydroxy-3(4-phenyl-1piperazinyl)]propyl-2,3-dihydro-6-methyl-1,3-dioxo-1H-pyrrolo[3,4-c]pyridine
P200
I. Muszalska
Stability of 4-methoxy-2-[2-hydroxy-3(4-phenyl-1-piperazinyl)]propyl-2,3-dihydro6-methyl-1,3-dioxo-1H-pyrrolo[3,4-c]pyridine in aqueous solutions
P201
B. Stanisz
The effect of humidity and temperature on the degradation of benazepril
hydrochloride (BEN)
P202
B. Stanisz
The stability of moexipril hydrochloride in solid phase
P203
B. Stanisz
Stability and mechanism of degradation of quinapril hydrochloride – mixture of
amorphous and crystalline forms (QHCl-AC) in solid phase
P204
A. Jelińska, L. Dobrowolski, I. Oszczapowicz
The stability of cefetamet pivoxil in aqueous solutions
P205
A. Jelińska, I. Dudzińska, I. Oszczapowicz
The kinetics of degradation of the amorphous form of cefuroxime axetil in solid
state
P206
M. Zając, A. Jelińska, J. Cielecka-Piontek, A. Kijewska, I. Oszczapowicz
Evaluation of the stability of aztreonam in solid state
P207
M. Zając, A. Jelińska, M. Sobczak, T. Wyrwicki, I. Oszczapowicz
The stability of daunorubicin hydrochloride in solid state
P208
L.I. Nadolnik, V.A. Basinsky
Preparation of thyroid gland organ culture, correction of experimental
hypothyroidism in rats
P209
N.M. Nasibullina, J.J. Sibgatullin, K.J. Sibgatullin
“VINIBIS this unique immunobiological product based"
P210
S. Busch, R. Gust
Transient transfection experiments on ERα and ERβ
P211
K. Majerz, B. Oleksyn, K. Stadnicka, J. Polański, H. Niedbała
Crystal structure of selected potential inhibitors of HIV-1 integrase
P212
A. Pioruńska-Mikołajczak, P. Mikołajczak, I. Okulicz-Kozaryn,
M. Pioruńska-Stolzmann, M. Iskra
Is acamprosate involved in lipid metabolism – study on outbred rats for high and
low ethanol preference
P213
Y. Martínez, V. Espinosa, S. Sepúlveda-Boza
Benzopyran-4-ones and its derivatives as inhibitors of human platelet
12-lipoxygenase
P214
J. Michálek, M. Přádný, J. Vacík, E. Peršínová, B. Dvořánková
Poly(methacrylate)s as polymer carriers for cultivation and transplantation of
keratinocytes onto large skin defects
P215
M. Pietsch, K. Taubert, B. Schulzeand, M. Gütschow
Inhibition of human leukocyte elastase by 2-phenylisothiazol-3(2H)-one
1,1-dioxides
P216
M. Bukowiecka–Matusiak, L.A. Woźniak, M.L. Navacchia, C. Chatgilialoglu
DNA damage. Synthesis and properties of oligonucleotides with incorporated
8-bromo-2’-deoxyadenosine and 5’,8-cyclo-2’-deoxyadenosine
P217
E. Forró F. Fülöp
Enzyme-catalyzed ring opening of cyclic and acyclicβ-lactams in organic solvent
P218
W. Sawuła, J. Jakóbkiewicz-Banecka, Z. Banecka-Majkutewicz, W. Nyka,
G. Węgrzyn, B. Banecki
Investigation of the influence of vitamin B6 on the total homocysteine level in blood
of stroke patients
P219
M. Pioruńska-Stolzmann, M. Iskra, W. Majewski, A. Pioruńska-Mikołajczak
Prostanoids as serum lipase inhibitors – the possible pharmacological applications
P220
B. Vanderhoydonck C.V. Stevens
Synthesis of 2-phosphonoaziridines from 1-phosphono-2-aza-1,3-dienes
P221
M. Teister, B. Czerny, E. Buszman
Modification of ovariectomy – induced disorders of biliary secretion by tamoxyfen
and raloxyfene
P222
H. Ekiert, U. Moroniewicz
Stationary liquid culture of Ruta graveolens L. shoots as a potential biotechnological
source of coumarins
P223
A. Szewczyk, H. Ekiert , E. Krystian
Conversion of hydroquinone to arbutin in shoot-differentiating callus culture of Ruta
graveolens ssp. divaricata (Tenore) Gams.
P224
A. Ptak, H. Ekiert, J. Gwiazda, E. Gomółka, A. Świderski, A. Bach
Optimization of light conditions for production of coumarins
in Ruta graveolens L. shoots cultivated in vitro